SCHEMBL3797930

SCHEMBL3797930

Fc1cccc(Cl)c1-c1ncc(-c2ccc(-c3noc(C4CCCC4)n3)nc2)[nH]1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGES O14684 4/20 0.46
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
ALDH1A1 P00352 1/20 0.43
TP53 P04637 1/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GRM5 P41594 4/20 0.39
PPARA Q07869 1/20 0.39
JAK2 O60674 1/20 0.38
DGAT1 O75907 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CNR2 P34972 1/20 0.38
CASP3 P42574 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
HPGDS O60760 1/20 0.37
HSD11B1 P28845 1/20 0.37
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3795318 0.99 PTGES (0.45) PTGESNPC1RAB9AALDH1A1TP53
SCHEMBL3796009 0.92 PTGES (0.44) PTGESNPC1RAB9AALDH1A1TP53
SCHEMBL3803620 0.91 PTGES (0.43) PTGESNPC1RAB9AALDH1A1TP53
SCHEMBL13076244 0.86 NPC1 (0.43) NPC1RAB9AALDH1A1TP53MAPK1
SCHEMBL13076236 0.86 NPC1 (0.45) NPC1RAB9AALDH1A1TP53MAPK1
SCHEMBL3790517 0.82 PTGES (0.54) PTGESNPC1RAB9AALDH1A1TP53
SCHEMBL3802070 0.81 PTGES (0.49) PTGESNPC1RAB9AJAK2L3MBTL1
SCHEMBL13076261 0.80 GRM5 (0.41) PTGESNPC1RAB9AALDH1A1TP53
SCHEMBL3797347 0.79 PTGES (0.50) PTGESNPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL3794424 0.79 PTGES (0.47) PTGESNPC1RAB9AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO claimed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed