SCHEMBL3796009

SCHEMBL3796009

Fc1cccc(Cl)c1-c1ncc(-c2ccc(-c3noc(C4CCC5(CC4)CC5)n3)nc2)[nH]1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGES O14684 4/20 0.44
GRM5 P41594 5/20 0.39
DGAT1 O75907 1/20 0.36
JAK2 O60674 1/20 0.36
CNR2 P34972 3/20 0.36
HPGDS O60760 3/20 0.36
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CNR1 P21554 2/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3803620 0.94 PTGES (0.43) PTGESGRM5DGAT1JAK2CNR2
SCHEMBL3797930 0.92 PTGES (0.46) PTGESGRM5DGAT1JAK2CNR2
SCHEMBL3795318 0.91 PTGES (0.45) PTGESGRM5DGAT1JAK2CNR2
SCHEMBL13076261 0.88 GRM5 (0.41) PTGESGRM5DGAT1CNR2NPC1
SCHEMBL13076379 0.81 GRM5 (0.45) GRM5DGAT1CNR2NPC1ALDH1A1
SCHEMBL3790517 0.80 PTGES (0.54) PTGESGRM5JAK2HPGDSNPC1
SCHEMBL3799989 0.80 PTGES (0.44) PTGESJAK2HPGDSNPC1RAB9A
SCHEMBL13076244 0.79 NPC1 (0.43) GRM5DGAT1CNR2NPC1ALDH1A1
SCHEMBL3802070 0.79 PTGES (0.49) PTGESJAK2HPGDSNPC1RAB9A
SCHEMBL13076236 0.78 NPC1 (0.45) GRM5DGAT1NPC1ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO claimed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed