SCHEMBL3802070

SCHEMBL3802070

CC(C)c1nc(-c2ccc(-c3cnc(-c4c(F)cccc4Cl)[nH]3)cn2)no1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 6/20 0.49
JAK2 O60674 1/20 0.42
HTT P42858 1/20 0.41
HPGDS O60760 5/20 0.41
NPC1 O15118 1/20 0.36
CASP3 P42574 1/20 0.36
RAB9A P51151 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA2 P47869 1/20 0.36
GABRA6 Q16445 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
NPY5R Q15761 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3794424 0.90 PTGES (0.47) PTGESJAK2HPGDSNPC1CASP3
SCHEMBL3793690 0.86 PTGES (0.46) PTGESJAK2HPGDSNPC1CASP3
SCHEMBL13076382 0.86 HTT (0.42) PTGESHTTNPC1CASP3RAB9A
SCHEMBL3790517 0.85 PTGES (0.54) PTGESJAK2HPGDSNPC1CASP3
SCHEMBL3797347 0.81 PTGES (0.50) PTGESJAK2HPGDSNPC1RAB9A
SCHEMBL3797930 0.81 PTGES (0.46) PTGESJAK2HPGDSNPC1CASP3
SCHEMBL3795318 0.80 PTGES (0.45) PTGESJAK2HPGDSNPC1CASP3
SCHEMBL3800503 0.80 PTGES (0.49) PTGESJAK2HPGDSNPC1RAB9A
SCHEMBL3803620 0.80 PTGES (0.43) PTGESJAK2HPGDSNPC1RAB9A
SCHEMBL3796009 0.79 PTGES (0.44) PTGESJAK2HPGDSNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO claimed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed