SCHEMBL13076261

SCHEMBL13076261

Fc1cccc(Cl)c1-c1nc(-c2ccc(-c3noc(C4CCC5(CC4)CC5)n3)nc2)c[nH]1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 10/20 0.41
DGAT1 O75907 1/20 0.38
CNR2 P34972 1/20 0.36
CHRNB2 P17787 2/20 0.35
CHRNA4 P43681 2/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PTGES O14684 1/20 0.34
HSD11B1 P28845 1/20 0.34
SMO Q99835 1/20 0.34
RORC P51449 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13076379 0.93 GRM5 (0.45) GRM5DGAT1CNR2CHRNB2CHRNA4
SCHEMBL13076244 0.91 NPC1 (0.43) GRM5DGAT1CNR2NPC1ALDH1A1
SCHEMBL13076236 0.91 NPC1 (0.45) GRM5DGAT1NPC1ALDH1A1TP53
SCHEMBL3796009 0.88 PTGES (0.44) GRM5DGAT1CNR2CHRNB2CHRNA4
SCHEMBL3803620 0.82 PTGES (0.43) GRM5DGAT1CNR2NPC1ALDH1A1
SCHEMBL3797930 0.80 PTGES (0.46) GRM5DGAT1CNR2NPC1ALDH1A1
SCHEMBL3795318 0.79 PTGES (0.45) GRM5DGAT1CNR2NPC1ALDH1A1
SCHEMBL13076233 0.79 RAB9A (0.43) GRM5NPC1ALDH1A1TP53MAPK1
SCHEMBL13076381 0.79 HSD11B1 (0.34) GRM5CHRNB2CHRNA4NPC1RAB9A
SCHEMBL13076382 0.78 HTT (0.42) CHRNB2CHRNA4NPC1ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed