SCHEMBL3800901

SCHEMBL3800901

O=C(NCc1c(Cl)cccc1Cl)c1cscn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK10 P53779 1/20 0.47
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
TSHR P16473 1/20 0.46
POLB P06746 1/20 0.46
GRM1 Q13255 1/20 0.44
ATM Q13315 1/20 0.43
GRM4 Q14833 2/20 0.43
HDAC3 O15379 2/20 0.43
HDAC1 Q13547 2/20 0.43
LMNA P02545 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
PIM1 P11309 1/20 0.42
MAP3K5 Q99683 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19476144 0.79 MMP13 (0.60) CYP1A2CYP2C19NPC1RAB9AALDH1A1
SCHEMBL4174785 0.77 SMN1; SMN2 (0.59) POLBLMNANPC1RAB9AALDH1A1
SCHEMBL29066497 0.75 CYP1A2 (0.48) MAPK10CYP1A2CYP3A4CYP2C19TSHR
SCHEMBL31703831 0.74 HDAC3 (0.42) CYP1A2CYP3A4CYP2C19TSHRGRM1
SCHEMBL29367205 0.73 HTT (0.69) TSHRPOLBLMNANPC1RAB9A
SCHEMBL3337029 0.73 KDM4E (0.50) TSHRPOLBGRM4HDAC3HDAC1
SCHEMBL28226304 0.73 MAP3K5 (0.52) GRM1GRM4HDAC3HDAC1LMNA
SCHEMBL29066486 0.72 NPC1 (0.53) MAPK10CYP1A2CYP3A4CYP2C19POLB
SCHEMBL29505784 0.72 SLC40A1 (0.48)
SCHEMBL29066483 0.72 NPC1 (0.53) MAPK10CYP1A2CYP3A4CYP2C19POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010114726-A1 AMINOBENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed