SCHEMBL3801722

SCHEMBL3801722

C=CC[Si](CC=C)(CC=C)CC(N)=O

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
FGFR4 P22455 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL175498 0.77 ABCC4 (0.34)
SCHEMBL2875011 0.70 TSHR (0.30) TSHR
SCHEMBL4563837 0.70 MCL1 (0.32) TSHR
SCHEMBL235304 0.67 TSHR (0.33) ALDH1A1TSHR
SCHEMBL9661307 0.65 ALOX15 (0.33) ALDH1A1
SCHEMBL7591793 0.65 ALDH1A1 (0.35) ALDH1A1TSHRFGFR4
SCHEMBL17201496 0.65 TSHR (0.31) ALDH1A1TSHR
SCHEMBL22988 0.64
SCHEMBL8064324 0.64 TSHR (0.41) TSHR
SCHEMBL9328869 0.63 ALDH1A1 (0.33) ALDH1A1TSHRFGFR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0273270-B1 PROCESS FOR THE PREPARATION OF (+)-BIOTIN LONZA AG (CH) 1992-04-08 EP claimed
EP-0270076-B1 IMIDAZOLE DERIVATIVES AND A PROCESS FOR THEIR PREPARATION LONZA AG (CH) 1991-10-09 EP claimed
EP-0299634-A2 Silicone polymer termination DOW CORNING CORPORATION (US) 1989-01-18 EP claimed
US-4766192-A MIXING POLYDIORGANOSILOXANE WITH PHOSPHORIC AND SILYLAMIDE COMPONENT DOW CORNING CORPORATION (US) 1988-08-23 US claimed
US-7825103-B2 5'-O-triisopropylsilyl-2'-cyano-2'-deoxy-1- beta -D-arabinofuranosylcytosine; antitumor agents TAIHO PHARMACEUTICAL CO., LTD. (JP) 2010-11-02 US disclosed
US-20090118222-A1 NOVEL PYRIMIDINE NUCLEOSIDE COMPOUND OR ITS SALT TAIHO PHARMACEUTICAL CO., LTD. (JP) 2009-05-07 US disclosed
EP-1845102-A1 NOVEL PYRIMIDINE NUCLEOSIDE COMPOUND OR ITS SALT TAIHO PHARMACEUTICAL COMPANY LIMITED (JP) 2007-10-17 EP disclosed
EP-1185365-A1 SURFACE-MODIFIED MIXED OXIDES CONTAINING PRECIOUS METAL AND TITANIUM, FOR THE SELECTIVE OXIDATION OF HYDROCARBONS Bayer Aktiengesellschaft (DE) 2002-03-13 EP disclosed
US-20010051754-A1 PLURAL STAGE TOLUENE DISPROPORTIONATION PROCESS MINIMIZING ETHYLBENZENE MOBIL OIL CORPORATION 2001-12-13 US disclosed
WO-2001009067-A1 PLURAL STAGE TOLUENE DISPROPORTIONATION PROCESS MINIMIZING ETHYLBENZENE PRODUCTION MOBIL OIL CORPORATION (US) 2001-02-08 WO disclosed
WO-2000064582-A1 SURFACE-MODIFIED MIXED OXIDES CONTAINING PRECIOUS METAL AND TITANIUM, FOR THE SELECTIVE OXIDATION OF HYDROCARBONS BAYER AKTIENGESELLSCHAFT (DE) 2000-11-02 WO disclosed
EP-0375040-A2 Process for the preparation of retro-inverso peptides and new intermediates thereof SCLAVO S.p.A. (IT) 1990-06-27 EP disclosed
US-4234721-A Process for the preparation of the crystalline monohydrate of 7-[D-amino-(p-hydroxyphenyl]acetamido)-3-methyl-3-cephen-4-carboxylic acid BRISTOL-MYERS COMPANY (US) 1980-11-18 US disclosed
US-4171431-A Nucleosides and process THE UPJOHN COMPANY (US) 1979-10-16 US disclosed
US-4160863-A ANTIBIOTIC BRISTOL-MYERS COMPANY (US) 1979-07-10 US disclosed
US-4066657-A ANTIBACTERIAL AGENTS FOR ANIMAL FEED SUPPLEMENTS PFIZER INC. (US) 1978-01-03 US disclosed
US-4036846-A ANTIBACTERIAL PFIZER INC. (US) 1977-07-19 US disclosed
US-4031077-A Antibacterial 3-phosphono penams PFIZER INC. (US) 1977-06-21 US disclosed
US-3994939-A BACTERICIDES PFIZER INC. (US) 1976-11-30 US disclosed
US-3943123-A ANTIBIOTIC KONINKLIJKE NEDERLANDSCHE GIST-EN SPIRITUSFABRIEK N.V. (NL) 1976-03-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090118222-A1 NOVEL PYRIMIDINE NUCLEOSIDE COMPOUND OR ITS SALT CDK10, SRSF9, SNRPD1 ALDH1A1 3707/4885TSHR 2261/4885FGFR4 2847/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.