SCHEMBL3814712

SCHEMBL3814712

CC1CCC(C(=O)N(c2cc(-c3cccc(C(F)(F)F)c3)sc2OC(=O)O)C(C)C)CC1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.37
AKR1C2 P52895 2/20 0.37
KMT2A Q03164 1/20 0.37
RXFP1 Q9HBX9 1/20 0.36
MCHR1 Q99705 1/20 0.36
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CCR2 P41597 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
JAK2 O60674 1/20 0.34
CNR2 P34972 1/20 0.34
S1PR5 Q9H228 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3816914 0.93 MMP1 (0.36) AKR1C3AKR1C2KMT2AMCHR1
SCHEMBL3807257 0.90 KDM4E (0.39) KMT2AALDH1A1SMN1; SMN2NPSR1TRPV1
SCHEMBL2879446 0.89 GRM5 (0.36) KMT2AJAK2
SCHEMBL2158041 0.88 ALDH1A1 (0.42) AKR1C3AKR1C2KMT2ARXFP1MCHR1
SCHEMBL3812117 0.88 HSD17B1 (0.39) NPSR1
SCHEMBL3814842 0.85 IKBKB (0.38) SMN1; SMN2NPSR1CYP1A2CYP2C19CNR2
SCHEMBL3809145 0.85 TRPV1 (0.38) KMT2AALDH1A1SMN1; SMN2NPSR1TRPV1
SCHEMBL3808993 0.84 MAPT (0.41) AKR1C3AKR1C2KMT2AALDH1A1
SCHEMBL3808983 0.84 MAPT (0.36) KMT2AALDH1A1NPSR1TRPV1
SCHEMBL3816814 0.83 KDM4E (0.39) KMT2AALDH1A1SMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401825-B1 THIOPHENE DERIVATIVES AS ANTIVIRAL AGENTS FOR FLAVIVIRUS INFECTION VIROCHEM PHARMA INC (CA) 2009-08-05 EP claimed