Leucine

Leucine

SCHEMBL3814957

CC(C)C[C@H](N)C(=O)O.O=C(O)[C@H](Cc1cccc2ccccc12)NS(=O)(=O)c1cccc2cccnc12.OB(O)O

nearest known ligand 0.45

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.45
ITGAV P06756 1/20 0.45
NTSR1 P30989 2/20 0.45
CYP3A4 P08684 3/20 0.44
CYP2C9 P11712 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2C19 P33261 2/20 0.44
MAPT P10636 2/20 0.44
GAA P10253 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
MMP1 P03956 1/20 0.43
ADAM17 P78536 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
HTR6 P50406 1/20 0.40
KCNH2 Q12809 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Leucine SCHEMBL1414045 0.97 ITGB3 (0.47) ITGB3ITGAVNTSR1CYP3A4CYP2C9
SCHEMBL232948 0.92 ITGB3 (0.45) ITGB3ITGAVNTSR1CYP3A4CYP2C9
Alanine SCHEMBL601223 0.90 ITGB3 (0.44) ITGB3ITGAVNTSR1CYP3A4CYP2C9
SCHEMBL3194343 0.86 ITGB3 (0.43) ITGB3ITGAVNTSR1CYP3A4CYP2C9
SCHEMBL31238101 0.83 PSMB5 (0.54) ITGB3ITGAVNTSR1CYP3A4CYP2C9
SCHEMBL7217344 0.82 MAPT (0.53) ITGB3ITGAVNTSR1CYP3A4CYP2C9
SCHEMBL5098994 0.80 NTSR1 (0.58) ITGB3ITGAVNTSR1CYP3A4CYP2C9
SCHEMBL5099014 0.80 NTSR1 (0.58) ITGB3ITGAVNTSR1CYP3A4CYP2C9
SCHEMBL7161574 0.78 NPSR1 (0.48) ITGB3ITGAVNTSR1CYP3A4CYP2C9
SCHEMBL1406185 0.78 GAA (0.38) ITGB3ITGAVNTSR1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0788360-B3 BORONIC ESTER AND ACID COMPOUNDS, SYNTHESIS AND USES MILLENNIUM PHARM INC (US) 2009-08-12 EP claimed
EP-1312609-B1 Boronic ester and acid compounds, synthesis and uses MILLENNIUM PHARM INC (US) 2005-12-28 EP claimed
EP-0788360-B1 BORONIC ESTER AND ACID COMPOUNDS, SYNTHESIS AND USES MILLENNIUM PHARM INC (US) 2003-05-28 EP claimed