SCHEMBL3815136

SCHEMBL3815136

COC(=O)Nc1cccc(CC(c2ccc(Cl)cc2)(c2cccnc2)c2ccnc(N)n2)n1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
NR2E3 Q9Y5X4 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
CYP3A4 P08684 2/20 0.37
CYP3A5 P20815 2/20 0.37
CYP19A1 P11511 5/20 0.36
PTGER2 P43116 1/20 0.34
GRM5 P41594 3/20 0.33
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1382291 0.78 NPC1 (0.37) KMT2ACYP19A1PTGER2GRM5SMN1; SMN2
SCHEMBL1381592 0.76 CYP19A1 (0.41) CYP3A4CYP3A5CYP19A1
SCHEMBL3813507 0.76 NAMPT (0.42) CYP3A4PTGER2GRM5
SCHEMBL1377766 0.76 CYP19A1 (0.49) CYP3A4CYP3A5CYP19A1
SCHEMBL3812181 0.75 LMNA (0.37) PTGER2
SCHEMBL3814798 0.73 CYP19A1 (0.43) CYP3A4CYP3A5CYP19A1PTGER2
SCHEMBL3811562 0.71 PTGER2 (0.38) PTGER2
SCHEMBL1379534 0.71 PTGER2 (0.36) PTGER2GRM5
SCHEMBL1379181 0.71 PTGER2 (0.36) PTGER2GRM5
SCHEMBL1377228 0.71 CYP1A2 (0.43) PTGER2GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776355-A4 POTASSIUM CHANNEL INHIBITORS MERCK & CO INC (US) 2009-08-12 EP disclosed
EP-1776355-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2007-04-25 EP disclosed
WO-2006014877-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2006-02-09 WO disclosed