SCHEMBL3815536

SCHEMBL3815536

COc1cccc(C(Cc2cccc(N)n2)(c2cccc(N)n2)c2cccc(OC)n2)n1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.39
MPO P05164 1/20 0.38
ADORA2A P29274 3/20 0.34
APP P05067 2/20 0.33
KDM1A O60341 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
MCHR1 Q99705 2/20 0.33
NOS2 P35228 2/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 2/20 0.32
IDH1 O75874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1381099 0.91 ADORA2A (0.35) BACE1MPOADORA2AAPPKDM1A
SCHEMBL3814663 0.84 BACE1 (0.33) BACE1MPOADORA2A
SCHEMBL1381051 0.76 NOS1 (0.38) MPONOS1
SCHEMBL331709 0.74
SCHEMBL29598348 0.74
SCHEMBL13830973 0.72 NOS2 (0.45) BACE1MPOAPPMCHR1NOS2
SCHEMBL15316717 0.71 KDM1A (0.43) MPOADORA2AKDM1AMAOAMAOB
SCHEMBL1377889 0.70 KCNA5 (0.36) BACE1APP
SCHEMBL1379821 0.70 NUDT1 (0.35)
SCHEMBL3812287 0.70 CYP19A1 (0.33) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776355-A4 POTASSIUM CHANNEL INHIBITORS MERCK & CO INC (US) 2009-08-12 EP disclosed
EP-1776355-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2007-04-25 EP disclosed
WO-2006014877-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2006-02-09 WO disclosed