SCHEMBL381593

SCHEMBL381593

CC(C)(C)N(C(=O)O)C(CNC=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.41
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.39
ACP3 P15309 2/20 0.39
CES2 O00748 1/20 0.39
GAA P10253 2/20 0.39
ATM Q13315 1/20 0.39
PNMT P11086 1/20 0.39
GPR139 Q6DWJ6 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRL1 P41146 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL381695 0.85 OPRM1 (0.43) BCHEALDH1A1MEN1CYP1A2POLB
SCHEMBL380987 0.83 ALDH1A1 (0.40) BCHEALDH1A1MEN1CYP1A2POLB
SCHEMBL15170368 0.83 ACP3 (0.47) ALDH1A1MEN1CYP1A2POLBCYP3A4
SCHEMBL381185 0.83 ACP3 (0.47) ALDH1A1MEN1CYP1A2POLBCYP3A4
SCHEMBL19244872 0.82 OPRM1 (0.48) BCHEALDH1A1MEN1CYP1A2POLB
SCHEMBL381880 0.82 SMN1; SMN2 (0.42) BCHEALDH1A1MEN1CYP1A2POLB
SCHEMBL16674214 0.82 PNMT (0.52) ALDH1A1MEN1CYP1A2POLBCYP3A4
SCHEMBL414657 0.82 ACP3 (0.43) ALDH1A1MEN1CYP1A2POLBCYP3A4
SCHEMBL19244815 0.79 ACP3 (0.40) ALDH1A1MEN1CYP1A2POLBCYP3A4
SCHEMBL19244817 0.78 KMT2A (0.41) ALDH1A1MEN1CYP1A2POLBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408751-B1 Substituted 2-acetamido-5-aryl-1,2,4-triazolones and use thereof BAYER IP GMBH (DE) 2017-08-23 EP disclosed
EP-2408751-A1 Substituted 2-acetamido-5-aryl-1,2,4-triazolones and use thereof Bayer Pharma Aktiengesellschaft (DE) 2012-01-25 EP disclosed
WO-2010105770-A1 SUBSTITUTED 2-ACETAMIDO-5-ARYL-1,2,4-TRIAZOLONES AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-09-23 WO disclosed