SCHEMBL3817562

SCHEMBL3817562

COc1ccc(C(C=O)Sc2ccc(Br)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.42
LMNA P02545 3/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
MAPT P10636 2/20 0.42
RAB9A P51151 2/20 0.42
MAPK1 P28482 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
ALDH1A1 P00352 3/20 0.41
SERPINH1 P50454 1/20 0.39
MAOA P21397 2/20 0.38
MAOB P27338 2/20 0.38
ADAM17 P78536 1/20 0.38
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
HTT P42858 1/20 0.37
CYP2A6 P11509 1/20 0.37
POLB P06746 1/20 0.37
IGF1R P08069 1/20 0.36
CYP1A1 P04798 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3818629 0.87 MEN1 (0.37) MEN1KMT2AMAOAMAOBCYP2A6
SCHEMBL20425444 0.83 MTNR1A (0.42) LMNAKMT2AMAPTRAB9AALDH1A1
SCHEMBL8057378 0.77 MAPT (0.50) NPSR1LMNAMEN1KMT2AMAPT
SCHEMBL9401376 0.72 L3MBTL1 (0.34) NPSR1LMNAMAPTRAB9AALDH1A1
SCHEMBL27907017 0.70 ALDH1A1 (0.50) NPSR1LMNAMEN1KMT2AMAPT
SCHEMBL9301 0.70
SCHEMBL14048314 0.69 MEN1 (0.52) NPSR1LMNAMEN1KMT2AMAPT
SCHEMBL7148548 0.69 NFE2L2 (0.44) KMT2ARAB9AALDH1A1MAOBNPC1
SCHEMBL9621498 0.68 ALDH1A1 (0.42) LMNAMEN1KMT2AMAPTRAB9A
Magnesium SCHEMBL31191739 0.68 CA1 (0.65) NPSR1LMNAMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2091527-A2 SULFIDE, SULFOXIDE AND SULFONE CHALCONE ANALOGUES, DERIVATIVES THEREOF AND THERAPEUTIC USES THEREOF Temple University of the Commonwealth System of Higher Education (US) 2009-08-26 EP disclosed
WO-2008076270-A2 SULFIDE, SULFOXIDE AND SULFONE CHALCONE ANALOGUES, DERIVATIVES THEREOF AND THERAPEUTIC USES THEREOF TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2008-06-26 WO disclosed