SCHEMBL381765

SCHEMBL381765

CC(C)(C)NOC(=O)CCNC(=O)c1ccc(N2CCC(Nc3ncccn3)CC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
GFER P55789 1/20 0.46
DRD2 P14416 7/20 0.43
DRD3 P35462 7/20 0.43
KDM4E B2RXH2 1/20 0.41
HTT P42858 1/20 0.41
CASR P41180 5/20 0.41
HPGDS O60760 1/20 0.41
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
JAK2 O60674 3/20 0.40
JAK1 P23458 2/20 0.40
JAK3 P52333 2/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40
HDAC1 Q13547 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6496334 0.91 CNR1 (0.43) DRD2DRD3KDM4EHTTCNR1
SCHEMBL6800155 0.90 ALDH1A1 (0.44) ALDH1A1GFERDRD2DRD3KDM4E
SCHEMBL7539445 0.89 CNR1 (0.44) ALDH1A1GFERDRD2DRD3KDM4E
SCHEMBL382963 0.88 SMYD3 (0.43) ALDH1A1GFERDRD2DRD3KDM4E
SCHEMBL6801441 0.87 ALDH1A1 (0.41) ALDH1A1GFERDRD2DRD3KDM4E
SCHEMBL383372 0.87 ITGB3 (0.42) JAK2JAK3
SCHEMBL381827 0.86 USP30 (0.45) DRD2DRD3
SCHEMBL382763 0.85 ITGB3 (0.48) GFERDRD2DRD3KDM4EHTT
SCHEMBL7540512 0.84 DRD2 (0.41) ALDH1A1GFERDRD2DRD3CASR
SCHEMBL382409 0.83 KDM4E (0.40) DRD2DRD3KDM4EHTTCASR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1074543-B1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA PHARMA CO LTD (JP) 2012-01-25 EP claimed
EP-1074543-B1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA PHARMA CO LTD (JP) 2012-01-25 EP disclosed