SCHEMBL3817754

SCHEMBL3817754

Cc1cccc(C)c1-c1nc(C)c(CN(CC(C)C)CC(C)C)c(N2C[CH]NCC2)n1

nearest known ligand 0.30

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
KMT2A Q03164 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3505822 0.83 C5AR1 (0.33) KDM4EALDH1A1LMNAGAAMAPT
SCHEMBL72878 0.78 JAK2 (0.33) KDM4EALDH1A1GAAKMT2A
SCHEMBL3509008 0.57 KDM4E (0.41) KDM4EALDH1A1LMNAGAAMAPT
SCHEMBL6186637 0.53 SLC6A2 (0.73) SLC6A2SLC6A4SLC6A3
SCHEMBL15855018 0.52 CHRM3 (0.39) KDM4EALDH1A1LMNAGAAKMT2A
SCHEMBL17532977 0.51 NOS3 (0.42) KDM4ELMNAGAAMAPT
SCHEMBL20110472 0.51 L3MBTL1 (0.50) ALDH1A1
SCHEMBL7354505 0.50 ADRB2 (0.60) ALDH1A1
SCHEMBL7773425 0.49 DRD2 (0.68) ALDH1A1LMNAGAAMAPT
SCHEMBL18176140 0.48 ACACB (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745033-A4 4,5-DISUBSTITUTED-2-ARYL PYRIMIDINES NEUROGEN CORP (US) 2009-08-26 EP claimed
EP-1745033-A2 4,5-DISUBSTITUTED-2-ARYL PYRIMIDINES NEUROGEN CORPORATION (US) 2007-01-24 EP claimed
WO-2005110416-A2 4,5-DISUBSTITUTED-2-ARYL PYRIMIDINES NEUROGEN CORPORATION (US) 2005-11-24 WO claimed