SCHEMBL381828

SCHEMBL381828

COc1cc(C(=O)NC(N)(CC(=O)O)C(C)(C)C)ccc1N1CCC(Nc2ncccn2)CC1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.43
DRD3 P35462 5/20 0.43
ITGB3 P05106 1/20 0.43
ITGAV P06756 1/20 0.43
ITGA2B P08514 1/20 0.43
USP30 Q70CQ3 2/20 0.41
EGFR P00533 2/20 0.38
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
NPY2R P49146 1/20 0.35
PTK2 Q05397 1/20 0.35
AURKA O14965 1/20 0.35
AURKB Q96GD4 1/20 0.35
SSTR4 P31391 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL383373 0.88 ITGB3 (0.40) ITGB3ITGAVITGA2BUSP30HDAC8
SCHEMBL381766 0.84 DRD2 (0.42) DRD2DRD3ITGB3ITGAVITGA2B
SCHEMBL382189 0.84 ITGB3 (0.50) DRD2DRD3ITGB3ITGAVITGA2B
SCHEMBL7650900 0.84 ITGB3 (0.44) DRD2DRD3ITGB3ITGAVITGA2B
SCHEMBL6496356 0.84 HDAC1 (0.41) DRD2DRD3
SCHEMBL382694 0.84 ITGB3 (0.46) DRD2DRD3ITGB3ITGAVITGA2B
SCHEMBL383236 0.83 ITGB3 (0.43) DRD2DRD3ITGB3ITGAVITGA2B
SCHEMBL383136 0.83 DRD2 (0.41) DRD2DRD3ITGB3ITGAVITGA2B
SCHEMBL383666 0.83 ITGB3 (0.46) DRD2DRD3ITGB3ITGAVITGA2B
SCHEMBL382101 0.82 ITGB3 (0.46) DRD2DRD3ITGB3ITGAVITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1074543-B1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA PHARMA CO LTD (JP) 2012-01-25 EP disclosed