SCHEMBL383136

SCHEMBL383136

COc1cc(C(=O)NC(CC(=O)O)(NC(=O)OCc2ccccc2)C(C)(C)C)ccc1N1CCC(Nc2ncccn2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41
ITGB3 P05106 2/20 0.41
ITGAV P06756 2/20 0.41
ITGA2B P08514 1/20 0.41
USP30 Q70CQ3 1/20 0.37
SMPD3 Q9NY59 1/20 0.37
HDAC1 Q13547 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
SMPD1 P17405 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
EHMT2 Q96KQ7 1/20 0.36
KDM1A O60341 2/20 0.35
MAOA P21397 2/20 0.35
KDM1B Q8NB78 2/20 0.35
RCOR1 Q9UKL0 2/20 0.35
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
ACHE P22303 2/20 0.35
PRMT5 O14744 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL382400 0.91 ITGB3 (0.38) ITGB3ITGAVITGA2BKDM1AMAOA
SCHEMBL381719 0.87 SYK (0.40) DRD2DRD3ITGB3ITGAVPRMT5
SCHEMBL6499250 0.87 VCP (0.40) DRD2DRD3ITGB3ITGAVHDAC1
SCHEMBL383138 0.86 ITGB3 (0.43) DRD2DRD3ITGB3ITGAVITGA2B
SCHEMBL382189 0.85 ITGB3 (0.50) DRD2DRD3ITGB3ITGAVITGA2B
SCHEMBL382988 0.84 PRMT5 (0.38) DRD2DRD3ITGB3ITGAVPRMT5
SCHEMBL381828 0.83 DRD2 (0.43) DRD2DRD3ITGB3ITGAVITGA2B
SCHEMBL382569 0.82 ITGB3 (0.43) DRD2DRD3ITGB3ITGAVITGA2B
SCHEMBL383666 0.82 ITGB3 (0.46) DRD2DRD3ITGB3ITGAVITGA2B
SCHEMBL382567 0.80 ITGB3 (0.55) ITGB3ITGAVITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1074543-B1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA PHARMA CO LTD (JP) 2012-01-25 EP disclosed