SCHEMBL3819367

SCHEMBL3819367

CCN(c1cccc(CN(c2ccc(F)cc2)[C@@H](C)C(N)=O)c1)C1CC1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.36
SLC6A2 P23975 4/20 0.35
SLC6A3 Q01959 4/20 0.35
SLC6A4 P31645 2/20 0.34
OPRM1 P35372 4/20 0.34
DPP4 P27487 2/20 0.34
DPP9 Q86TI2 2/20 0.34
DPP7 Q9UHL4 2/20 0.34
OPRD1 P41143 2/20 0.34
OPRK1 P41145 2/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
GRIA2 P42262 1/20 0.33
GRIN2A Q12879 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
UBE2M P61081 1/20 0.33
DCUN1D1 Q96GG9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3817654 0.82 CYP3A4 (0.37) DPP4DPP9DPP7UBE2MDCUN1D1
SCHEMBL3819363 0.82 ATM (0.39) S1PR1SLC6A2SLC6A3OPRM1DPP4
SCHEMBL3821795 0.81 GRIN2A (0.41) S1PR1SLC6A2SLC6A3SLC6A4OPRM1
SCHEMBL3821794 0.80 OPRM1 (0.39) S1PR1OPRM1MAOA
SCHEMBL3059109 0.79 ACHE (0.39) S1PR1SLC6A2SLC6A3SLC6A4OPRM1
Hydrochloric Acid SCHEMBL3064216 0.78 ACHE (0.39) S1PR1SLC6A2SLC6A3SLC6A4OPRM1
SCHEMBL3819801 0.77 ATM (0.40) OPRM1DPP4DPP9DPP7OPRD1
SCHEMBL3819226 0.76 CNR1 (0.40) OPRM1UBE2MDCUN1D1
SCHEMBL3064159 0.76 CHRM1 (0.42)
SCHEMBL13090640 0.75 S1PR1 (0.38) S1PR1SLC6A2SLC6A3SLC6A4OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2091917-A1 ION CHANNEL MODULATORS Wyeth a Corporation of the State of Delaware (US) 2009-08-26 EP claimed
WO-2008073934-A1 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed