SCHEMBL3821795

SCHEMBL3821795

CCN(c1cccc(CN(CC(N)=O)c2ccc(F)cc2)c1)C1CC1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRIN2A Q12879 6/20 0.41
GRIA2 P42262 5/20 0.41
KDM1A O60341 2/20 0.37
S1PR1 P21453 2/20 0.36
PTPN1 P18031 1/20 0.36
SLC6A2 P23975 3/20 0.35
SLC6A4 P31645 3/20 0.35
SLC6A3 Q01959 3/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
SSTR3 P32745 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
F2 P00734 1/20 0.34
F10 P00742 1/20 0.34
PRSS1 P07477 1/20 0.34
PRSS2 P07478 1/20 0.34
PRSS3 P35030 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3821794 0.82 OPRM1 (0.39) S1PR1OPRM1
SCHEMBL3819367 0.81 S1PR1 (0.36) GRIN2AGRIA2S1PR1SLC6A2SLC6A4
SCHEMBL3819363 0.79 ATM (0.39) S1PR1SLC6A2SLC6A3OPRM1
SCHEMBL3059109 0.79 ACHE (0.39) S1PR1SLC6A2SLC6A4SLC6A3OPRM1
Hydrochloric Acid SCHEMBL3064216 0.78 ACHE (0.39) S1PR1SLC6A2SLC6A4SLC6A3OPRM1
SCHEMBL3064159 0.77 CHRM1 (0.42) KDM1A
SCHEMBL13090640 0.77 S1PR1 (0.38) GRIN2AGRIA2S1PR1SLC6A2SLC6A4
SCHEMBL4734946 0.76 LMNA (0.58) OPRM1
SCHEMBL3819801 0.76 ATM (0.40) OPRM1OPRD1OPRK1
SCHEMBL3819014 0.75 CNR2 (0.46) CNR1CNR2OPRM1F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2091917-A1 ION CHANNEL MODULATORS Wyeth a Corporation of the State of Delaware (US) 2009-08-26 EP claimed
WO-2008073934-A1 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed