SCHEMBL382074

SCHEMBL382074

CC(C)(C)C(CC(=O)O)(NC(=O)c1ccc(N2CCN(Cc3nc4ccccc4[nH]3)CC2)cc1)NS(=O)(=O)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 16/20 0.51
NPC1 O15118 1/20 0.50
GAA P10253 1/20 0.50
HTR1A P08908 1/20 0.46
ADRA2C P18825 1/20 0.46
HTR2A P28223 1/20 0.46
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
DRD2 P14416 2/20 0.43
DRD3 P35462 1/20 0.43
CYP3A4 P08684 1/20 0.41
ALOX15 P16050 1/20 0.41
OPRK1 P41145 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
GLA P06280 1/20 0.41
MAPT P10636 1/20 0.41
ATM Q13315 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL382571 0.84 ITGB3 (0.42) NPC1GAAKDM4EALDH1A1TDP1
SCHEMBL382076 0.83 DRD4 (0.51) DRD4NPC1GAAHTR1AADRA2C
SCHEMBL415668 0.80 DRD4 (0.54) DRD4NPC1GAAHTR1AADRA2C
SCHEMBL415667 0.77 ITGB3 (0.64) DRD4NPC1GAAHTR1AADRA2C
SCHEMBL460323 0.76 ITGB3 (0.41) TDP1GLAMAPTATM
SCHEMBL7655325 0.75 DRD4 (0.52) DRD4NPC1GAAHTR1AADRA2C
SCHEMBL383213 0.75 DRD4 (0.77) DRD4NPC1GAAHTR1AADRA2C
SCHEMBL383159 0.75 ITGB3 (0.44) KDM4ETDP1DRD2DRD3GLA
SCHEMBL382073 0.74 DRD4 (0.49) DRD4NPC1GAAHTR1AADRA2C
SCHEMBL382075 0.73 ITGB3 (0.50) DRD4NPC1GAAHTR1AADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1074543-B1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA PHARMA CO LTD (JP) 2012-01-25 EP disclosed