SCHEMBL382075

SCHEMBL382075

CC(C)(C)c1ccccc1S(=O)(=O)N[C@@H](CNC(=O)c1ccc(N2CCN(Cc3nc4ccccc4[nH]3)CC2)cc1)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.50
ITGA2B P08514 3/20 0.50
DRD4 P21917 9/20 0.49
NPC1 O15118 1/20 0.48
GAA P10253 1/20 0.48
HTR1A P08908 1/20 0.44
ADRA2C P18825 1/20 0.44
HTR2A P28223 1/20 0.44
ITGAV P06756 7/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
ITGA2 P17301 1/20 0.42
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL415667 0.89 ITGB3 (0.64) ITGB3ITGA2BDRD4NPC1GAA
SCHEMBL382572 0.84 ITGAV (0.53) ITGB3ITGA2BITGAVITGA2
SCHEMBL7651216 0.78 ITGB3 (0.68) ITGB3ITGA2BITGAV
SCHEMBL460324 0.77 ITGAV (0.53) ITGB3ITGA2BITGAVITGA2
SCHEMBL382076 0.76 DRD4 (0.51) DRD4NPC1GAAHTR1AADRA2C
SCHEMBL383160 0.75 ITGAV (0.58) ITGB3ITGA2BITGAVITGA2
SCHEMBL383468 0.74 ITGB3 (0.51) ITGB3ITGA2BITGAVITGA2
SCHEMBL383213 0.73 DRD4 (0.77) DRD4NPC1GAAHTR1AADRA2C
SCHEMBL415668 0.73 DRD4 (0.54) ITGB3ITGA2BDRD4NPC1GAA
SCHEMBL6500394 0.73 ITGAV (0.50) ITGB3ITGA2BITGAVKDM4EITGA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1074543-B1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA PHARMA CO LTD (JP) 2012-01-25 EP disclosed