SCHEMBL3821050

SCHEMBL3821050

COc1cc2c(cc1F)CNC=C2

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.37
BRD4 O60885 1/20 0.36
DRD5 P21918 4/20 0.33
CYP3A4 P08684 1/20 0.31
MAPT P10636 1/20 0.31
KDM1A O60341 2/20 0.31
ALDH1A1 P00352 1/20 0.31
NCOA1 Q15788 1/20 0.31
NCOA3 Q9Y6Q9 1/20 0.31
TDP2 O95551 1/20 0.31
LMNA P02545 1/20 0.30
MAPK1 P28482 1/20 0.30
HTT P42858 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL525652 0.86 CYP3A4 (0.45) PARP1BRD4CYP3A4MAPTALDH1A1
Hydrochloric Acid SCHEMBL4762831 0.84 PARP1 (0.44) PARP1BRD4CYP3A4MAPTALDH1A1
SCHEMBL11045652 0.75 GAA (0.57) BRD4DRD5CYP3A4MAPTALDH1A1
SCHEMBL11041542 0.75 BRD4 (0.38) BRD4DRD5CYP3A4MAPTALDH1A1
SCHEMBL19038489 0.69 GAA (0.58) PARP1DRD5MAPTALDH1A1MAPK1
SCHEMBL10650554 0.69 MAOA (0.45) BRD4CYP3A4MAPTALDH1A1LMNA
SCHEMBL29561779 0.69 MAOA (0.45) BRD4CYP3A4MAPTALDH1A1LMNA
SCHEMBL2937347 0.66 LMNA (0.46) CYP3A4MAPTKDM1ALMNAMAPK1
SCHEMBL11043204 0.66 BRD4 (0.44) BRD4DRD5CYP3A4MAPTALDH1A1
SCHEMBL4807201 0.65 BRD4 (0.40) BRD4MAPTALDH1A1LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2089385-A2 INHIBITORS OF HEPATITIS C VIRUS Brystol-Myers Squibb Company (US) 2009-08-19 EP disclosed
EP-2086967-A2 INHIBITORS OF HEPATITIS C VIRUS Brystol-Myers Squibb Company (US) 2009-08-12 EP disclosed
WO-2008057871-A2 INHIBITORS OF HEPATITIS C VIRUS BRISTOL-MYERS SQUIBB COMPANY (US) 2008-05-15 WO disclosed
WO-2008057873-A2 INHIBITORS OF HEPATITIS C VIRUS BRISTOL-MYERS SQUIBB COMPANY (US) 2008-05-15 WO disclosed