SCHEMBL3822003

SCHEMBL3822003

CCN(c1ccccc1O)C1CCN(C(C)CCNC(=O)OC(C)(C)C)CC1

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 8/20 0.41
UBE2M P61081 11/20 0.41
DCUN1D1 Q96GG9 11/20 0.41
DRD2 P14416 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4598395 0.76 GPR119 (0.51)
SCHEMBL3757285 0.75 IDO1 (0.44) CCR5DRD2
SCHEMBL3757286 0.75 IDO1 (0.44) CCR5DRD2
SCHEMBL13052234 0.73 KMT2A (0.43) DRD2
SCHEMBL3757466 0.72 CCR5 (0.41) CCR5DRD2
SCHEMBL4240911 0.72 CCR5 (0.65) CCR5
SCHEMBL3768194 0.72 UBE2M (0.47) UBE2MDCUN1D1
SCHEMBL3768190 0.72 UBE2M (0.47) UBE2MDCUN1D1
SCHEMBL3764142 0.72 CCR5 (0.39) CCR5DRD2
SCHEMBL4240711 0.70 CCR5 (0.60) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942890-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORP (US) 2009-08-26 EP disclosed
EP-1942890-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2008-07-16 EP disclosed
WO-2006138350-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-12-28 WO disclosed