SCHEMBL38239

SCHEMBL38239

COc1cnc(-c2[c]cccc2)cn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OXTR P30559 14/20 0.35
AVPR1A P37288 5/20 0.35
SIRT6 Q8N6T7 1/20 0.34
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA5 P31644 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33
GABRB2 P47870 1/20 0.33
GABRA4 P48169 1/20 0.33
GABRE P78334 1/20 0.33
GABRA6 Q16445 1/20 0.33
GABRG1 Q8N1C3 1/20 0.33
GABRG3 Q99928 1/20 0.33
GABRQ Q9UN88 1/20 0.33
CYP2A6 P11509 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38536 0.77 CYP2A6 (0.49) OXTRCYP2A6NPC1
SCHEMBL38086 0.76 LMNA (0.38) NPC1RAB9AKDM4E
SCHEMBL28477929 0.74 TDP1 (0.30)
SCHEMBL17504866 0.72 ALOX5AP (0.38) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL714399 0.70 CCR1 (0.54) CYP2A6NPC1RAB9AKDM4E
SCHEMBL28986650 0.70 TRPV4 (0.35)
SCHEMBL715526 0.69
SCHEMBL17504881 0.69 IDO1 (0.41) GABRA1GABRG2GABRB3
SCHEMBL2185307 0.69 BACE1 (0.37) OXTRAVPR1ASIRT6NPC1RAB9A
SCHEMBL3138241 0.68 SIRT6 (0.56) SIRT6GABRPGABRDGABRA1GABRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011151436-A2 NOVEL COMPOUNDS, METHOD FOR USE THEM AND PHARMACEUTICAL COMPOSITION CONTAINING THEM EUROSCREEN S.A. (BE) 2011-12-08 WO disclosed