SCHEMBL382649

SCHEMBL382649

C#C[C@@H](NC(=O)c1ccc(N2CCC(Nc3ncccn3)CC2)cc1)C(CC)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.41
ITGAV P06756 3/20 0.41
ITGA2B P08514 3/20 0.41
ITGB1 P05556 2/20 0.41
ITGA5 P08648 2/20 0.41
ITGB5 P18084 2/20 0.41
DRD2 P14416 7/20 0.40
DRD3 P35462 7/20 0.40
CASR P41180 4/20 0.40
CHRNA7 P36544 1/20 0.37
CHRNA10 Q9GZZ6 1/20 0.37
CHRNA9 Q9UGM1 1/20 0.37
DGAT1 O75907 1/20 0.37
JAK2 O60674 1/20 0.36
HDAC1 Q13547 1/20 0.36
JAK1 P23458 1/20 0.36
SMYD3 Q9H7B4 1/20 0.36
USP2 O75604 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL382117 0.82 DRD2 (0.44) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL6796559 0.78 CASR (0.45) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL383016 0.78 DRD2 (0.55) DRD2DRD3CASRUSP2
SCHEMBL382964 0.77 CASR (0.45) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL6796240 0.76 DRD2 (0.43) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL6796554 0.76 ITGB3 (0.49) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL382962 0.75 ITGB3 (0.49) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL28747046 0.75 ITGB3 (0.49) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL6800173 0.74 CASR (0.43) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL6796225 0.74 CASR (0.44) ITGB3ITGAVITGA2BDRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1074543-B1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA PHARMA CO LTD (JP) 2012-01-25 EP disclosed