SCHEMBL382990

SCHEMBL382990

CC(C)(C)[C@@](CNC(=O)c1ccc(N2CCC(Nc3ncccn3)CC2)c(F)c1F)(NC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 4/20 0.38
ITGAV P06756 4/20 0.38
PRMT5 O14744 1/20 0.35
GRIN2B Q13224 3/20 0.35
FKBP1A P62942 2/20 0.34
SYK P43405 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
TRPA1 O75762 1/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
CTSK P43235 1/20 0.33
GAA P10253 1/20 0.32
RORC P51449 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA2A P29274 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL382402 0.88 ITGB3 (0.40) ITGB3ITGAVGRIN2BALDH1A1LMNA
SCHEMBL382988 0.85 PRMT5 (0.38) ITGB3ITGAVPRMT5GRIN2BSYK
SCHEMBL383138 0.84 ITGB3 (0.43) ITGB3ITGAVDRD2DRD3
SCHEMBL381721 0.84 ITGB3 (0.40) ITGB3ITGAVPRMT5GRIN2BSYK
SCHEMBL382802 0.83 ITGB3 (0.37) ITGB3ITGAVALDH1A1DRD2DRD3
SCHEMBL6499269 0.82 VCP (0.40) ITGB3ITGAVGRIN2BSYKALDH1A1
SCHEMBL382611 0.82 ITGB3 (0.47) ITGB3ITGAV
SCHEMBL382612 0.80 GAA (0.37) ITGB3ITGAVPRMT5GRIN2BSYK
SCHEMBL382613 0.79 ITGB3 (0.42) ITGB3ITGAVPRMT5GRIN2B
SCHEMBL382989 0.79 ITGB3 (0.36) ITGB3ITGAVPRMT5GRIN2BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1074543-B1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA PHARMA CO LTD (JP) 2012-01-25 EP disclosed