SCHEMBL3835967

SCHEMBL3835967

O=C(O)c1ccc(C#Cc2cccnc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.61
MKNK1 Q9BUB5 1/20 0.57
MKNK2 Q9HBH9 1/20 0.57
ALDH1A1 P00352 1/20 0.56
APP P05067 1/20 0.56
GAA P10253 1/20 0.56
HCAR3 P49019 1/20 0.56
HCAR2 Q8TDS4 1/20 0.56
HAO1 Q9UJM8 2/20 0.53
RARB P10826 1/20 0.49
RARG P13631 1/20 0.49
CYP2A6 P11509 3/20 0.47
HIF1A Q16665 2/20 0.47
EPAS1 Q99814 2/20 0.47
PTPN11 Q06124 1/20 0.46
KMO O15229 1/20 0.46
CYP2E1 P05181 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C9 P11712 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29908914 0.85 ALDH1A1 (0.55) FFAR1MKNK1MKNK2ALDH1A1APP
SCHEMBL29603820 0.83 KMO (0.59) FFAR1MKNK1MKNK2ALDH1A1APP
SCHEMBL16720129 0.83 KMO (0.59) FFAR1MKNK1MKNK2ALDH1A1APP
SCHEMBL13907278 0.83 CYP2A6 (0.62) FFAR1CYP2A6CYP2E1CYP3A4CYP2D6
SCHEMBL400670 0.82 HDAC1 (0.60) FFAR1HIF1AEPAS1
SCHEMBL28718553 0.82 KMO (0.58) FFAR1MKNK1MKNK2ALDH1A1APP
SCHEMBL402518 0.81 RARB (0.62) FFAR1APPRARBRARGPTPN11
SCHEMBL401836 0.81 GRM5 (0.64) FFAR1APPCYP2A6CYP2E1CYP3A4
SCHEMBL31673222 0.81 GRM5 (0.64) FFAR1APPCYP2A6CYP2E1CYP3A4
SCHEMBL3838348 0.81 ALDH1A1 (0.61) FFAR1ALDH1A1HAO1CYP2A6HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1729771-B1 PYRIDYL DERIVATIVES AND THEIR USE AS MGLU5 RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2009-10-14 EP claimed