SCHEMBL3838348

SCHEMBL3838348

COC(=O)c1ccc(C#Cc2cccnc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.61
FFAR1 O14842 1/20 0.52
PTPN11 Q06124 1/20 0.51
CYP19A1 P11511 1/20 0.50
CYP11B1 P15538 1/20 0.50
CYP11B2 P19099 1/20 0.50
SLC2A1 P11166 1/20 0.50
CSF1R P07333 1/20 0.49
KMT2A Q03164 1/20 0.48
HIF1A Q16665 1/20 0.46
EPAS1 Q99814 1/20 0.46
CYP2A6 P11509 1/20 0.46
CYP2C9 P11712 1/20 0.46
CHRNB2 P17787 1/20 0.46
CYP2B6 P20813 1/20 0.46
CYP2C19 P33261 1/20 0.46
CHRNA4 P43681 1/20 0.46
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HAO1 Q9UJM8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3719847 0.86 ALDH1A1 (0.52) ALDH1A1FFAR1CYP19A1CYP11B1CYP11B2
SCHEMBL3714223 0.85 ALDH1A1 (0.62) ALDH1A1CYP19A1CYP11B1CYP11B2SLC2A1
SCHEMBL3712736 0.85 ALDH1A1 (0.62) ALDH1A1CYP19A1CYP11B1CYP11B2CSF1R
SCHEMBL3710033 0.84 ALDH1A1 (0.54) ALDH1A1FFAR1CYP19A1CYP11B1CYP11B2
SCHEMBL22833769 0.83 CSF1R (0.68) ALDH1A1CYP19A1CYP11B1CYP11B2SLC2A1
SCHEMBL3714187 0.82 ALDH1A1 (0.51) ALDH1A1FFAR1CYP19A1CYP11B1CYP11B2
SCHEMBL25210061 0.82 PTPN11 (0.58) ALDH1A1FFAR1PTPN11CYP2C9CYP2C19
SCHEMBL1105504 0.82 TSHR (0.67) ALDH1A1PTPN11KMT2ACYP2C9CYP2C19
SCHEMBL69268 0.82 PTPN11 (0.69) ALDH1A1PTPN11KMT2ACYP2C9CYP2C19
SCHEMBL29506324 0.82 CSF1R (0.53) ALDH1A1CYP19A1CYP11B1CYP11B2SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1729771-B1 PYRIDYL DERIVATIVES AND THEIR USE AS MGLU5 RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2009-10-14 EP claimed
EP-1729771-B1 PYRIDYL DERIVATIVES AND THEIR USE AS MGLU5 RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2009-10-14 EP disclosed