SCHEMBL3837307

SCHEMBL3837307

Cc1ccccc1NCc1cc(I)c2c(c1)CNC2=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 3/20 0.44
ADRA2B P18089 1/20 0.42
MAPT P10636 5/20 0.36
HTT P42858 2/20 0.36
HDAC8 Q9BY41 3/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
KDM4E B2RXH2 3/20 0.35
MEN1 O00255 2/20 0.35
ALDH1A1 P00352 2/20 0.35
KMT2A Q03164 2/20 0.35
PDE4B Q07343 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CRHBP P24387 1/20 0.33
CYP2C19 P33261 1/20 0.33
CRHR2 Q13324 1/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3836956 0.75 SLC2A1 (0.35)
SCHEMBL3835531 0.71 GSR (0.35) ALDH1A1KDRPDGFRB
SCHEMBL3837309 0.71 PARP1 (0.40) HDAC1MEN1KMT2ACRHBPCRHR2
SCHEMBL3836776 0.70 AURKA (0.34) KDM4EKDR
SCHEMBL3839397 0.70 PDGFRB (0.33) KDRPDGFRB
SCHEMBL3835406 0.70 PARP1 (0.45)
SCHEMBL3839331 0.70 KDR (0.32) KDR
SCHEMBL3834548 0.68 NAMPT (0.39) HDAC1KDM4ECYP3A4LMNA
SCHEMBL3839251 0.68 PARP1 (0.33) HTTHDAC8HDAC6HPGD
SCHEMBL3836958 0.68 PARP1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2108642-A1 JAK INHIBITOR Kyowa Hakko Kirin Co., Ltd. (JP) 2009-10-14 EP disclosed