SCHEMBL3710033

SCHEMBL3710033

COC(=O)c1cncc(-c2ccc(C#Cc3cccnc3)cc2)c1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.54
CYP11B1 P15538 2/20 0.51
CYP11B2 P19099 2/20 0.51
CYP19A1 P11511 1/20 0.51
SLC2A1 P11166 1/20 0.48
XDH P47989 1/20 0.46
NEK1 Q96PY6 1/20 0.46
FFAR1 O14842 1/20 0.44
MKNK1 Q9BUB5 1/20 0.44
MKNK2 Q9HBH9 1/20 0.44
NR4A2 P43354 1/20 0.44
ATM Q13315 1/20 0.43
CYP2A6 P11509 1/20 0.43
AAK1 Q2M2I8 2/20 0.43
CSF1R P07333 1/20 0.43
HAO1 Q9UJM8 1/20 0.42
ERN1 O75460 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3714223 0.87 ALDH1A1 (0.62) ALDH1A1CYP11B1CYP11B2CYP19A1SLC2A1
SCHEMBL13188366 0.86 CYP11B1 (0.67) ALDH1A1CYP11B1CYP11B2CYP19A1SLC2A1
SCHEMBL3838348 0.84 ALDH1A1 (0.61) ALDH1A1CYP11B1CYP11B2CYP19A1SLC2A1
SCHEMBL3713649 0.84 HDAC1 (0.52) XDHFFAR1MKNK1MKNK2AAK1
SCHEMBL31704881 0.83 ALDH1A1 (0.68) ALDH1A1CYP11B1CYP11B2CYP19A1SLC2A1
SCHEMBL29771391 0.83 ALDH1A1 (0.68) ALDH1A1CYP11B1CYP11B2CYP19A1SLC2A1
SCHEMBL3714867 0.83 ALDH1A1 (0.68) ALDH1A1CYP11B1CYP11B2CYP19A1SLC2A1
SCHEMBL31705350 0.83 ALDH1A1 (0.68) ALDH1A1CYP11B1CYP11B2CYP19A1SLC2A1
SCHEMBL3712340 0.82 CYP11B2 (0.53) ALDH1A1CYP11B1CYP11B2XDHMKNK1
SCHEMBL10028685 0.82 ALDH1A1 (0.66) ALDH1A1CYP11B1CYP11B2CYP19A1SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed