SCHEMBL3839402

SCHEMBL3839402

CN(Cc1cc(I)c2c(c1)CNC2=O)C1CCCCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.43
HRH4 Q9H3N8 1/20 0.43
PARP1 P09874 4/20 0.38
CYP2D6 P10635 2/20 0.36
ABCB11 O95342 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
AR P10275 1/20 0.36
SLC6A2 P23975 1/20 0.36
PDE4A P27815 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
KCNH2 Q12809 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
LMNA P02545 2/20 0.36
CYP3A4 P08684 1/20 0.36
HTT P42858 1/20 0.36
LTA4H P09960 2/20 0.34
ALDH1A1 P00352 3/20 0.34
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3839251 0.77 PARP1 (0.33) HRH3PARP1HTT
SCHEMBL3839331 0.71 KDR (0.32)
SCHEMBL3836956 0.70 SLC2A1 (0.35) PARP1
SCHEMBL3837343 0.69 L3MBTL1 (0.39) PARP1HTTALDH1A1MAPTSMN1; SMN2
SCHEMBL3834414 0.69 PARP1 (0.48) HRH3HRH4PARP1ALDH1A1SMN1; SMN2
SCHEMBL3837163 0.67 KDR (0.35)
SCHEMBL2393018 0.65 HRH3 (0.74) HRH3HRH4PARP1CYP2D6ABCB11
SCHEMBL11593176 0.65 CYP2D6 (0.71) HRH3HRH4PARP1CYP2D6ABCB11
SCHEMBL3836136 0.64 PARP1 (0.31) PARP1
SCHEMBL3835531 0.64 GSR (0.35) ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2108642-A1 JAK INHIBITOR Kyowa Hakko Kirin Co., Ltd. (JP) 2009-10-14 EP disclosed