SCHEMBL3839795

SCHEMBL3839795

COc1c(OC(N)=O)[nH]c2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.53
ALDH1A1 P00352 3/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
KMT2A Q03164 3/20 0.44
HPGD P15428 2/20 0.44
HSD17B10 Q99714 2/20 0.44
MEN1 O00255 2/20 0.44
NR4A2 P43354 2/20 0.44
GSK3B P49841 2/20 0.43
ADK P55263 2/20 0.43
TUBB4A P04350 5/20 0.43
TUBB P07437 5/20 0.43
TUBA3C P0DPH7 5/20 0.43
TUBA1B P68363 5/20 0.43
TUBA4A P68366 5/20 0.43
TUBB4B P68371 5/20 0.43
TUBB3 Q13509 5/20 0.43
TUBB2A Q13885 5/20 0.43
TUBB8 Q3ZCM7 5/20 0.43
TUBA3E Q6PEY2 5/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6526599 0.87 GSK3B (0.56) KDM4EALDH1A1SMN1; SMN2KMT2AHPGD
SCHEMBL3839803 0.86 TUBB4A (0.44) KDM4EALDH1A1SMN1; SMN2KMT2AHPGD
SCHEMBL3838681 0.84 KIF11 (0.42) KDM4EALDH1A1SMN1; SMN2KMT2AHPGD
SCHEMBL3837499 0.84 HTR6 (0.41) KDM4EALDH1A1SMN1; SMN2KMT2AHPGD
SCHEMBL3836337 0.84 KDM4E (0.41) KDM4EALDH1A1SMN1; SMN2KMT2AHPGD
SCHEMBL3839787 0.82 SCN9A (0.43) KDM4EALDH1A1KMT2AHPGDHSD17B10
SCHEMBL9573791 0.80 TUBB4A (0.46) KDM4EALDH1A1SMN1; SMN2KMT2AHPGD
SCHEMBL4208427 0.79 KDM4E (0.51) KDM4EALDH1A1SMN1; SMN2KMT2AHPGD
SCHEMBL3835352 0.79 HSD17B10 (0.48) KDM4EALDH1A1KMT2AHPGDHSD17B10
SCHEMBL2348968 0.78 MAP2 (0.55) KDM4EALDH1A1SMN1; SMN2KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1791537-B1 3-ARYLTHIOINDOLE-2-CARBOXAMIDE DERIVATIVES AND ANALOGS THEREOF AS INHIBITORS OF CASEIN KINASE I AVENTIS PHARMA INC (US) 2009-10-14 EP claimed