SCHEMBL3844004

SCHEMBL3844004

CCCCC=C(c1ccc(O)cc1)c1ccc(O)cc1

nearest known ligand 0.62

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 15/20 0.62
ESR2 Q92731 15/20 0.62
HSD17B3 P37058 5/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8622933 0.92 ESR1 (0.64) ESR1ESR2HSD17B3
SCHEMBL16685069 0.88 ESR1 (0.50) ESR1ESR2HSD17B3
SCHEMBL2566604 0.82 HSD17B3 (0.47) ESR1ESR2HSD17B3
SCHEMBL11994148 0.82 HTR7 (0.50) ESR1ESR2
SCHEMBL2566602 0.82 HSD17B3 (0.47) ESR1ESR2HSD17B3
SCHEMBL6897257 0.82 SIGMAR1 (0.54) ESR1ESR2
SCHEMBL16685238 0.82 ESR1 (0.46) ESR1ESR2
SCHEMBL14288468 0.81 ESR1 (0.50) ESR1ESR2
SCHEMBL16685139 0.80 ESR1 (0.44) ESR1ESR2
SCHEMBL16684967 0.80 TBXAS1 (0.51) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951217-A4 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2009-08-12 EP claimed
EP-1951217-A2 CHEMICAL COMPOUNDS SmithKline Beecham Corporation (US) 2008-08-06 EP claimed
WO-2007062148-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-05-31 WO claimed
EP-3063158-A1 METALLOCENE DERIVATIVES WITH ANTICANCER ACTIVITY Paris Sciences et Lettres - Quartier Latin (FR) 2016-09-07 EP disclosed
WO-2015063201-A1 METALLOCENE DERIVATIVES WITH ANTICANCER ACTIVITY PARIS SCIENCES ET LETTRES - QUARTIER LATIN (FR) 2015-05-07 WO disclosed