SCHEMBL3846952

SCHEMBL3846952

COc1cc(F)c2cc(CC=O)c(=O)[nH]c2c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.36
KDM4E B2RXH2 10/20 0.35
ALDH1A1 P00352 8/20 0.35
HSD17B10 Q99714 6/20 0.34
TSHR P16473 4/20 0.34
TRAP1 Q12931 1/20 0.34
GAA P10253 3/20 0.34
MAPT P10636 3/20 0.34
NPSR1 Q6W5P4 3/20 0.34
ALOX15 P16050 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
APAF1 O14727 1/20 0.34
NPC1 O15118 1/20 0.34
MAPK1 P28482 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
HPGD P15428 2/20 0.33
LMNA P02545 2/20 0.33
MEN1 O00255 1/20 0.33
HCRTR1 O43613 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3841830 0.81 GRIN1 (0.36) KDM4E
SCHEMBL3843000 0.78 GRIN1 (0.39) KDM4EALDH1A1HSD17B10SMN1; SMN2NPC1
SCHEMBL3846232 0.75 KDM4E (0.56) KDM4EALDH1A1HSD17B10TSHRGAA
SCHEMBL3839869 0.74 DAO (0.56) KDM4EALDH1A1HSD17B10MAPTNPC1
SCHEMBL2461361 0.72 TAAR1 (0.55) TAAR1ALDH1A1TRAP1
SCHEMBL3840529 0.69 PARP1 (0.45) KDM4EALDH1A1MEN1KMT2A
SCHEMBL3864985 0.69 KDM4E (0.57) KDM4EALDH1A1HSD17B10GAAMAPT
SCHEMBL4438609 0.68 CHRM2 (0.47) ALDH1A1
SCHEMBL14992582 0.66 TAAR1 (0.47) TAAR1ALDH1A1TRAP1MAPTSMN1; SMN2
SCHEMBL21490329 0.66 ULK1 (0.53) KDM4EALDH1A1HSD17B10GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044077-A1 DERIVATIVES AND ANALOGS OF N-ETHYLQUINOLONES AND N-ETHYLAZAQUINOLONES Glaxo Group Limited (GB) 2009-04-08 EP disclosed
WO-2008009700-A1 DERIVATIVES AND ANALOGS OF N-ETHYLQUINOLONES AND N-ETHYLAZAQUINOLONES GLAXO GROUP LIMITED (GB) 2008-01-24 WO disclosed