SCHEMBL384749

SCHEMBL384749

COC(=O)c1cc(Cl)c(N)cc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 1.00
KDM4E B2RXH2 1/20 0.64
HTR4 Q13639 4/20 0.60
CYP3A4 P08684 2/20 0.60
CYP1A2 P05177 2/20 0.60
CYP2D6 P10635 2/20 0.60
HTR3A P46098 2/20 0.60
CYP2C9 P11712 1/20 0.60
TSHR P16473 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
GLA P06280 1/20 0.56
NPC1 O15118 1/20 0.56
HTT P42858 1/20 0.56
HTR3E A5X5Y0 1/20 0.56
SLC22A1 O15245 1/20 0.56
HTR3B O95264 1/20 0.56
ALDH1A1 P00352 1/20 0.56
LMNA P02545 1/20 0.56
MPO P05164 1/20 0.56
ADRA2A P08913 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7405359 0.98 GAA (0.97) GAAKDM4EHTR4CYP3A4CYP1A2
SCHEMBL31321292 0.91 GAA (0.82) GAAKDM4EHTR4CYP3A4CYP1A2
SCHEMBL8292456 0.88 GAA (0.79) GAAKDM4EHTR4CYP3A4CYP1A2
SCHEMBL7853424 0.86 GAA (0.76) GAAKDM4EHTR4CYP3A4CYP1A2
SCHEMBL7419408 0.85 GAA (0.74) GAAKDM4ESMN1; SMN2GLANPC1
SCHEMBL6473999 0.85 GAA (0.74) GAAKDM4EHTR4CYP3A4CYP1A2
SCHEMBL29424850 0.85 GAA (0.74) GAAKDM4EHTR4CYP3A4CYP1A2
SCHEMBL9379986 0.85 GAA (0.74) GAAHTR4CYP3A4CYP1A2CYP2D6
SCHEMBL725809 0.84 GAA (0.73) GAAHTR4CYP3A4CYP1A2CYP2D6
SCHEMBL7280230 0.84 GAA (0.73) GAAHTR4CYP3A4CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 229 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12606523-B2 Deuterated organic compounds and uses thereof ENGRAIL THERAPEUTICS, INC. (US) 2026-04-21 US disclosed
CN-119977828-A Methoxychlor-pup Process for the preparation of amines 河南优凯制药有限公司 2025-05-13 CN disclosed
CN-119977827-A Methoxychlor-pram intermediate and preparation method and application thereof 河南优凯制药有限公司 2025-05-13 CN disclosed
US-20250091990-A1 DEUTERATED ORGANIC COMPOUNDS AND USES THEREOF ENGRAIL THERAPEUTICS, INC. 2025-03-20 US disclosed
US-20250041319-A1 BICYCLIC HETEROARYL DERIVATIVES AS ECTONUCLEOTIDE PYROPHOSPHATASE PHOSPHODIESTERASE 1 INHIBITORS RIBOSCIENCE LLC 2025-02-06 US disclosed
US-20250011280-A1 DEUTERATED ORGANIC COMPOUNDS AND USES THEREOF ENGRAIL THERAPEUTICS, INC. 2025-01-09 US disclosed
EP-4460292-A1 DEUTERATED ORGANIC COMPOUNDS AND USES THEREOF Engrail Therapeutics, Inc. (US) 2024-11-13 EP disclosed
EP-4460490-A1 DEUTERATED ORGANIC COMPOUNDS AND USES THEREOF Engrail Therapeutics, Inc. (US) 2024-11-13 EP disclosed
CN-118804910-A Deuterated organic compounds and use thereof 恩格雷尔治疗有限公司 2024-10-18 CN disclosed
CN-118804746-A Deuterated organic compounds and use thereof 恩格雷尔治疗有限公司 2024-10-18 CN disclosed
US-5063230-A Substituted saturated and unsaturated indole quinoline and benzazepine carboxamides and their use as pharmacological agents RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-11-05 US disclosed
WO-1991004738-A1 DIBENZOFURANCARBOXAMIDES RORER INTERNATIONAL (HOLDINGS), INC. (US) 1991-04-18 WO disclosed
US-4959485-A 5-HT3 ANTAGONISTS RORER PHARMACEUTICAL CORPORATION (US) 1990-09-25 US disclosed
WO-1990006113-A1 SUBSTITUTED SATURATED AND UNSATURATED INDOLE QUINOLINE AND BENZAZEPINE CARBOXAMIDES AND THEIR USE AS PHARMACOLOGICAL AGENTS RORER INTERNATIONAL (OVERSEAS) INC. (US) 1990-06-14 WO disclosed
US-4920219-A Substituted saturated and unsaturated indole quinoline and benzazepine carboxamides and their use as pharmacological agents RORER PHARMACEUTICAL CORP. (US) 1990-04-24 US disclosed
US-4914117-A ANTIDEPRESSANTS, CENTRAL NERVOUS SYSTEM ACTIVATORS; DOPAMINE ANTAGONISTS SOCIETE D'ETUDES SCIENTIFIQUES ET INDUSTRIELLE DE L'ILE-D-FRANCE (FR) 1990-04-03 US disclosed
WO-1989010364-A1 DIBENZOFURANCARBOXAMIDES RORER INTERNATIONAL (OVERSEAS) INC. (US) 1989-11-02 WO disclosed
EP-0339950-A2 Dibenzofurancarboxamides, their use as pharmaceutical agents, a composition containing the same, and a process for the preparation thereof RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1989-11-02 EP disclosed
US-4863921-A Dibenzofurancarboxamides and their pharmaceutical compositions and methods RORER PHARMACEUTICAL CORPORATION (US) 1989-09-05 US disclosed
US-4835172-A Novel benzamides, intermediates and process for the preparation and therapeutic use thereof SOCIETE D'ETUDES SCIENTIFIQUES ET INDUSTRIELLES DE L'ILE-DE-FRANCE (FR) 1989-05-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250041319-A1 BICYCLIC HETEROARYL DERIVATIVES AS ECTONUCLEOTIDE PYROPHOSPHATASE PHOSPHODIESTERASE 1 INHIBITORS ENPP1, ENPP3, SMPD1 GAA 154/4885KDM4E 2905/4885HTR4 4266/4885
US-20250091990-A1 DEUTERATED ORGANIC COMPOUNDS AND USES THEREOF DRD1, DRD4, DRD2 GAA 2151/4885KDM4E 3482/4885HTR4 13/4885
US-12606523-B2 Deuterated organic compounds and uses thereof DRD1, DRD2, DRD3 GAA 4676/4885KDM4E 3058/4885HTR4 37/4885
US-20250011280-A1 DEUTERATED ORGANIC COMPOUNDS AND USES THEREOF DBH, DRD1, OPRD1 GAA 1451/4885KDM4E 3024/4885HTR4 68/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.