SCHEMBL4715804

SCHEMBL4715804

Cc1ccnc(NC(=O)c2ccc(-c3cnc4ccc(-c5cn[nH]c5)cn34)cc2F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.43
PTK6 Q13882 1/20 0.41
AURKB Q96GD4 1/20 0.41
FLT3 P36888 2/20 0.41
NRAS P01111 1/20 0.41
MAP3K5 Q99683 1/20 0.41
SORT1 Q99523 2/20 0.41
CLK1 P49759 2/20 0.41
CLK2 P49760 2/20 0.41
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
CHEK1 O14757 5/20 0.39
KIT P10721 1/20 0.39
CHEK2 O96017 1/20 0.39
ABL1 P00519 1/20 0.39
PKM P14618 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GRM5 P41594 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3847724 0.99 LOXL2 (0.42) LOXL2PTK6AURKBFLT3NRAS
Hydrochloric Acid SCHEMBL4715592 0.89 SORT1 (0.43) PTK6AURKBFLT3NRASMAP3K5
SCHEMBL3856718 0.89 NPC1 (0.46) PTK6AURKBFLT3NRASMAP3K5
Hydrochloric Acid SCHEMBL5852371 0.88 NPC1 (0.45) PTK6AURKBFLT3NRASMAP3K5
Hydrochloric Acid SCHEMBL4717129 0.86 LOXL2 (0.41) LOXL2SORT1NPC1RAB9APKM
Hydrochloric Acid SCHEMBL3846519 0.86 KIT (0.43) PTK6AURKBFLT3NRASMAP3K5
Hydrochloric Acid SCHEMBL3849166 0.84 FLT3 (0.42) PTK6AURKBFLT3NRASMAP3K5
SCHEMBL3846729 0.84 SMN1; SMN2 (0.46) FLT3NRASMAP3K5SORT1CLK1
SCHEMBL4713522 0.83 CHEK1 (0.42) PTK6AURKBFLT3NRASMAP3K5
Hydrochloric Acid SCHEMBL3847294 0.83 SMN1; SMN2 (0.45) FLT3NRASMAP3K5SORT1CLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP claimed