SCHEMBL3875112

SCHEMBL3875112

COc1cccc(NC(C)CSC)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
MAPT P10636 2/20 0.48
GAA P10253 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
KCNH3 Q9ULD8 1/20 0.48
ALDH1A1 P00352 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
MAPK1 P28482 1/20 0.45
POLB P06746 1/20 0.45
MTNR1B P49286 4/20 0.45
MTNR1A P48039 3/20 0.45
TSHR P16473 1/20 0.43
RAPGEF4 Q8WZA2 1/20 0.43
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21790727 0.83 ALDH1A1 (0.52) MEN1KMT2AMAPTGAANPSR1
SCHEMBL9781352 0.82 ALDH1A1 (0.51) MEN1KMT2AMAPTGAANPSR1
SCHEMBL17604272 0.82 MAPT (0.49) MEN1KMT2AMAPTGAANPSR1
SCHEMBL631776 0.79 KCNH3 (0.64) MEN1KMT2AMAPTKCNH3ALDH1A1
Hydrochloric Acid SCHEMBL2249099 0.78 KCNH3 (0.67) MEN1KMT2AMAPTKCNH3ALDH1A1
SCHEMBL2704334 0.77 TSHR (0.53) MEN1KMT2AALDH1A1POLBMTNR1B
SCHEMBL28885886 0.76 KCNH3 (0.53) MEN1KMT2AMAPTKCNH3ALDH1A1
SCHEMBL10989610 0.76 KCNH3 (0.53) MEN1KMT2AMAPTGAAKCNH3
SCHEMBL2918668 0.75 TDP1 (0.54) GAANPSR1KCNH3ALDH1A1L3MBTL1
SCHEMBL3650245 0.73 MTNR1A (0.41) MEN1KMT2AMAPTGAANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118076-A1 QUINOXALINE COMPOUNDS AND USE THEREOF Merck Serono S.A. (CH) 2009-11-18 EP disclosed
WO-2008101979-A1 QUINOXALINE COMPOUNDS AND USE THEREOF MERCK SERONO S.A. (CH) 2008-08-28 WO disclosed