SCHEMBL3877875

SCHEMBL3877875

CCOC(=O)NN=C(Cc1cccnc1C(F)(F)F)c1cc(OCc2ccccc2)c(OCc2ccccc2)c([N+](=O)[O-])c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
PKM P14618 1/20 0.40
HPGD P15428 1/20 0.40
PTGES O14684 1/20 0.39
MAPT P10636 3/20 0.35
NPC1 O15118 1/20 0.35
NFKB1 P19838 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
PPIA P62937 4/20 0.35
CTSV O60911 3/20 0.35
CTSL P07711 3/20 0.35
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.34
PPIF P30405 1/20 0.34
MYC P01106 1/20 0.34
MAX P61244 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3877870 1.00 SMN1; SMN2 (0.40) SMN1; SMN2PKMHPGDPTGESMAPT
SCHEMBL3586711 0.92 PTGES (0.42) PTGESMAPTNPC1RAB9APPIA
SCHEMBL3586707 0.92 PTGES (0.42) PTGESMAPTNPC1RAB9APPIA
SCHEMBL3586703 0.92 PTGES (0.42) PTGESMAPTNPC1RAB9APPIA
SCHEMBL1447461 0.85 PTGES (0.40) SMN1; SMN2PKMHPGDPTGESMAPT
SCHEMBL3587958 0.83 PPIA (0.41) PTGESMAPTNPC1RAB9APPIA
SCHEMBL4942728 0.81 SMN1; SMN2 (0.37) SMN1; SMN2PKMHPGDPTGESMAPT
SCHEMBL30105376 0.74 RAB9A (0.46) SMN1; SMN2PKMPTGESMAPTNPC1
SCHEMBL3593506 0.74 CTSV (0.42) PTGESMAPTNPC1RAB9APPIA
SCHEMBL3593504 0.73 NPC1 (0.45) SMN1; SMN2PKMPTGESMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2027091-A1 NEW PHARMACEUTICAL COMPOUNDS BIAL - Portela & Ca., S.A. (PT) 2009-02-25 EP disclosed
WO-2007117165-A1 NEW PHARMACEUTICAL COMPOUNDS BIAL - PORTELA & CA, S.A. (PT) 2007-10-18 WO disclosed