SCHEMBL4942728

SCHEMBL4942728

CCOC(=O)NN=C(CC1=C(C(F)(F)F)N=CCC1=O)c1cc(OCc2ccccc2)c(OCc2ccccc2)c([N+](=O)[O-])c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.37
PKM P14618 2/20 0.37
HPGD P15428 1/20 0.37
PTGES O14684 1/20 0.37
MAPT P10636 3/20 0.33
ALDH1A1 P00352 1/20 0.33
CTSV O60911 3/20 0.33
CTSL P07711 3/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
MYC P01106 1/20 0.32
MAX P61244 1/20 0.32
ABCB1 P08183 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ELANE P08246 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4947748 0.85 PTGES (0.38) PTGESMAPTCTSVCTSLKDM4E
SCHEMBL3877870 0.81 SMN1; SMN2 (0.40) SMN1; SMN2PKMHPGDPTGESMAPT
SCHEMBL3877875 0.81 SMN1; SMN2 (0.40) SMN1; SMN2PKMHPGDPTGESMAPT
SCHEMBL1447461 0.78 PTGES (0.40) SMN1; SMN2PKMHPGDPTGESMAPT
SCHEMBL3586711 0.73 PTGES (0.42) PTGESMAPTALDH1A1CTSVCTSL
SCHEMBL3586707 0.73 PTGES (0.42) PTGESMAPTALDH1A1CTSVCTSL
SCHEMBL3586703 0.73 PTGES (0.42) PTGESMAPTALDH1A1CTSVCTSL
SCHEMBL4948554 0.67 EIF4E (0.38) SMN1; SMN2MAPTKDM4EABCB1CYP19A1
SCHEMBL13257189 0.67 LMNA (0.61) SMN1; SMN2HPGDPTGESMAPTCTSV
SCHEMBL1447206 0.67 CTSV (0.55) PTGESMAPTCTSVCTSLMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907382-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS Portela & C.A. S.A (PT) 2008-04-09 EP disclosed
WO-2007013830-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS PORTELA & CA. S.A. (PT) 2007-02-01 WO disclosed