SCHEMBL3878440

SCHEMBL3878440

Cc1c(Cc2ccccc2C(=O)O)cc(-c2ccc(Cl)cc2Cl)c(-c2ccc(Br)cc2)[n+]1[O-]

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 4/20 0.39
DHODH Q02127 1/20 0.37
DCLRE1B Q9H816 1/20 0.36
POLB P06746 1/20 0.35
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34
MARS1 P56192 2/20 0.34
SRD5A2 P31213 1/20 0.33
LTB4R2 Q9NPC1 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
CNR1 P21554 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3878435 1.00 MRGPRX4 (0.39) MRGPRX4DHODHDCLRE1BPOLBALDH1A1
SCHEMBL3878437 0.81 DHODH (0.38) MRGPRX4DHODHPOLBALDH1A1TP53
SCHEMBL4514869 0.81 RAB9A (0.40) POLBALDH1A1CNR1
SCHEMBL4513890 0.65 DHODH (0.38) DHODHMARS1SRD5A2
SCHEMBL4505429 0.65 DHODH (0.50) DHODHALDH1A1TP53SRD5A2CNR1
SCHEMBL442223 0.64 ALDH1A1 (0.58) MRGPRX4ALDH1A1TP53SRD5A2CA1
SCHEMBL16950095 0.62 TSHR (0.72) ALDH1A1CA1CA2CA9
SCHEMBL5455142 0.61 ALDH1A1 (0.61) MRGPRX4ALDH1A1TP53
SCHEMBL27853748 0.61 ALDH1A1 (0.61) MRGPRX4ALDH1A1TP53SRD5A2CA1
SCHEMBL69352 0.61 TSHR (0.68) POLBALDH1A1TP53CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010492-A2 AMINOMETHYL PYRIDINE DERIVATIVES, METHOD FOR PREPARING SAME AND THERAPEUTIC USE THEREOF Sanofi-Aventis (FR) 2009-01-07 EP disclosed
WO-2007119001-A2 AMINOMETHYL PYRIDINE DERIVATIVES, METHOD FOR PREPARING SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2007-10-25 WO disclosed