SCHEMBL3878583

SCHEMBL3878583

CS(=O)(=O)c1ccc(C2CCN(C(=O)O)CC2)cc1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QDPR P09417 2/20 0.44
THRA P10827 1/20 0.43
VDR P11473 1/20 0.43
THRB P10828 1/20 0.43
SLC9A1 P19634 4/20 0.41
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
DRD2 P14416 2/20 0.38
GPR119 Q8TDV5 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
DRD3 P35462 2/20 0.36
HTR6 P50406 2/20 0.36
HRH3 Q9Y5N1 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16262649 0.82 HDAC1 (0.49) QDPRHDAC3HDAC1HDAC2CA12
SCHEMBL3871895 0.81 THRB (0.60) THRAVDRTHRB
SCHEMBL3871890 0.81 THRB (0.60) THRAVDRTHRB
SCHEMBL23122328 0.79 QDPR (0.56) QDPRHDAC3HDAC1HDAC2CA12
SCHEMBL12478958 0.78 QDPR (0.48) QDPRHDAC3HDAC1HDAC2HRH3
SCHEMBL3817499 0.78 QDPR (0.44) QDPRHDAC3HDAC1HDAC2
SCHEMBL14624308 0.77 GPR119 (0.51) QDPRTHRAVDRTHRBCA12
SCHEMBL23122840 0.76 QDPR (0.56) QDPRHDAC3HDAC1HDAC2CA12
SCHEMBL16318326 0.76 QDPR (0.43) QDPRHDAC3HDAC1HDAC2CA12
SCHEMBL12479689 0.76 QDPR (0.46) QDPRHDAC3HDAC1HDAC2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115393-A1 PROCESS FOR THE PREPARATION OF N-(1-PHENYLETHYL)ANILINES, SALTS, AND SOLVATES THEREOF USEFUL AS SEROTONIN 5-HT6 ANTAGONISTS LABORATORIOS DEL DR. ESTEVE, S. A. (ES) 2009-09-24 WO disclosed
EP-2103596-A1 Process for the preparation of N-(phenylethyl) anilines salts and solvates thereof useful as serotonin 5-HT6 antagonists Laboratorios Del. Dr. Esteve, S.A. (ES) 2009-09-23 EP disclosed