SCHEMBL3871895

SCHEMBL3871895

CS(=O)(=O)c1ccc(C2CCN(C(=O)O)CC2)cc1[N+](=O)[O-]

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
THRB P10828 16/20 0.60
THRA P10827 5/20 0.60
VDR P11473 1/20 0.60
VCAM1 P19320 1/20 0.47
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3871890 1.00 THRB (0.60) THRBTHRAVDRVCAM1POLB
SCHEMBL3869166 0.87 THRB (0.55) THRBTHRAVDR
SCHEMBL3878583 0.81 QDPR (0.44) THRBTHRAVDR
SCHEMBL4184466 0.78 THRB (0.57) THRBTHRAVDR
SCHEMBL22095447 0.78 THRB (0.59) THRBTHRAVDRVCAM1
SCHEMBL14624308 0.77 GPR119 (0.51) THRBTHRAVDR
SCHEMBL853823 0.74 SLC18A3 (0.58)
SCHEMBL4440176 0.71 HCAR3 (0.54) POLB
SCHEMBL4440170 0.71 HCAR3 (0.54) POLB
SCHEMBL3530451 0.70 VCAM1 (0.71) THRBTHRAVCAM1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115393-A1 PROCESS FOR THE PREPARATION OF N-(1-PHENYLETHYL)ANILINES, SALTS, AND SOLVATES THEREOF USEFUL AS SEROTONIN 5-HT6 ANTAGONISTS LABORATORIOS DEL DR. ESTEVE, S. A. (ES) 2009-09-24 WO disclosed
EP-2103596-A1 Process for the preparation of N-(phenylethyl) anilines salts and solvates thereof useful as serotonin 5-HT6 antagonists Laboratorios Del. Dr. Esteve, S.A. (ES) 2009-09-23 EP disclosed