SCHEMBL3888484

SCHEMBL3888484

O=C(N[C@@H]1N=C(c2ccccc2)c2ccccc2N(CC(F)(F)F)C1=O)Oc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.59
CCKBR P32239 1/20 0.53
CALCRL Q16602 14/20 0.52
RAMP1 O60894 2/20 0.49
SENP1 Q9P0U3 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9423126 0.84 CCKBR (0.74) CCKBR
SCHEMBL9422961 0.84 CCKBR (0.74) CCKBR
SCHEMBL9422957 0.84 CCKBR (0.74) CCKBR
SCHEMBL4410860 0.80 KCNH2 (0.54) KCNH2CCKBRSENP1
SCHEMBL8223082 0.78 KCNH2 (0.73) KCNH2CALCRLRAMP1
SCHEMBL3252895 0.77 KCNH2 (0.47) KCNH2CCKBRCALCRLRAMP1
SCHEMBL4413834 0.76 SENP1 (0.56) CCKBRSENP1
SCHEMBL9866235 0.76 CCKBR (0.59) CCKBR
SCHEMBL7212286 0.75 KCNH2 (0.64) KCNH2CCKBRCALCRLRAMP1
SCHEMBL9256656 0.75 CCKBR (0.40) CCKBRSENP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1856100-A4 CGRP RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2009-04-15 EP disclosed
EP-1856100-A2 CGRP RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2007-11-21 EP disclosed
WO-2006078554-A2 CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2006-07-27 WO disclosed