SCHEMBL390989

SCHEMBL390989

CCC(N)c1ccc(Cl)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.57
ADRB2 P07550 1/20 0.56
SLC6A3 Q01959 4/20 0.45
SLC6A2 P23975 2/20 0.45
SCN4A P35499 2/20 0.44
AOC3 Q16853 2/20 0.42
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
TSHR P16473 2/20 0.41
MAPK1 P28482 2/20 0.41
HIF1A Q16665 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
LMNA P02545 2/20 0.39
TP53 P04637 1/20 0.39
HPGD P15428 1/20 0.39
KDM4E B2RXH2 1/20 0.39
RAB9A P51151 1/20 0.39
MEN1 O00255 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1977034 1.00 SLC6A4 (0.57) SLC6A4ADRB2SLC6A3SLC6A2SCN4A
SCHEMBL12262253 1.00 SLC6A4 (0.57) SLC6A4ADRB2SLC6A3SLC6A2SCN4A
Hydrochloric Acid SCHEMBL16292773 0.98 SLC6A4 (0.55) SLC6A4ADRB2SLC6A3SLC6A2SCN4A
SCHEMBL23092069 0.87 SLC6A4 (0.70) SLC6A4ADRB2SLC6A3SLC6A2SCN4A
SCHEMBL8284225 0.83 SLC6A4 (0.59) SLC6A4ADRB2SLC6A3SLC6A2IDO1
SCHEMBL8285910 0.83 SLC6A4 (0.59) SLC6A4ADRB2SLC6A3SLC6A2IDO1
SCHEMBL9198692 0.82 ADRB2 (0.52) SLC6A4ADRB2SLC6A3SLC6A2SCN4A
Hydrochloric Acid SCHEMBL4938618 0.81 SLC6A4 (0.57) SLC6A4ADRB2IDO1MAPK1HIF1A
Hydrochloric Acid SCHEMBL4935308 0.81 SLC6A4 (0.57) SLC6A4ADRB2IDO1MAPK1HIF1A
Ammonia Solution, Strong SCHEMBL386864 0.80 ADRB2 (0.50) SLC6A4ADRB2SLC6A3SLC6A2SCN4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3994125-B1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF REGENERON PHARMA (US) 2025-12-24 EP disclosed
US-12252495-B2 Protein kinase B inhibitors ASTRAZENECA AB (SE) 2025-03-18 US disclosed
US-20240299402-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF REGENERON PHARMACEUTICALS, INC. (US) 2024-09-12 US disclosed
US-11957687-B2 Modulators of HSD17B13 and methods of use thereof REGENERON PHARMACEUTICALS, INC. (US) 2024-04-16 US disclosed
US-20240109902-A1 PROTEIN KINASE B INHIBITORS ASTRAZENECA AB (SE) 2024-04-04 US disclosed
US-11760760-B2 Protein kinase B inhibitors ASTRAZENECA AB (SE) 2023-09-19 US disclosed
US-20230094341-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF REGENERON PHARMACEUTICALS, INC. (US) 2023-03-30 US disclosed
US-20220220116-A1 PROTEIN KINASE B INHIBITORS ASTRAZENECA AB (SE) 2022-07-14 US disclosed
EP-3994125-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF Regeneron Pharmaceuticals, Inc. (US) 2022-05-11 EP disclosed
US-11236095-B2 Protein kinase B inhibitors ASTRAZENECA AB (SE) 2022-02-01 US disclosed
WO-2005090348-A1 PYRAZOLO ’3,4-B! PYRIDINE COMPOUNDS, AND THEIR USE AS PHOSPHODIESTERASE TYPE 4 (PDE4) INHIBITORS GLAXO GROUP LIMITED (GB) 2005-09-29 WO disclosed
WO-2005058892-A1 PYRAZOLO [3,4-B] PYRIDINE COMPOUNDS, AND THEIR USE AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LIMITED (GB) 2005-06-30 WO disclosed
EP-1373192-A1 N-PHENPROPYLCYCLOPENTYL-SUBSTITUTED GLUTARAMIDE DERIVATIVES AS NEP INHIBITORS FOR FSAD Pfizer Limited (GB) 2004-01-02 EP disclosed
WO-2002079143-A1 N-PHENPROPYLCYCLOPENTYL-SUBSTITUTED GLUTARAMIDE DERIVATIVES AS NEP INHIBITORS FOR FSAD PFIZER LIMITED (GB) 2002-10-10 WO disclosed
US-5017723-A Psychotropic Agents JOUVEINAL S.A. (FR) 1991-05-21 US disclosed
EP-0210044-B1 HYDROXY AND ALKOXY PYRIMIDINES PFIZER INC. (US) 1990-08-29 EP disclosed
US-4711888-A Hydroxy and alkoxy pyrimidines PFIZER INC. (US) 1987-12-08 US disclosed
EP-0210044-A2 Hydroxy and alkoxy pyrimidines PFIZER INC. (US) 1987-01-28 EP disclosed
US-4622324-A CARDIOVASCULAR DISORDERS, HYPOTENSIVES DR. WILLMAR SCHWABE GMBH & CO. (DE) 1986-11-11 US disclosed
US-4479951-A CORONARY DIESASE DR. WILLMAR SCHWABE GMBH & CO. (DE) 1984-10-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12252495-B2 Protein kinase B inhibitors PRKAR2B, PRKCB, AKT1 SLC6A4 4654/4885ADRB2 1451/4885SLC6A3 4750/4885
US-20220220116-A1 PROTEIN KINASE B INHIBITORS PRKAR2B, PRKCB, AKT1 SLC6A4 4654/4885ADRB2 1451/4885SLC6A3 4750/4885
US-20240299402-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF HSD17B3, HSD17B11, HSD17B1 SLC6A4 2816/4885ADRB2 1854/4885SLC6A3 2221/4885
US-20240109902-A1 PROTEIN KINASE B INHIBITORS PRKAR2B, PRKCB, AKT1 SLC6A4 4654/4885ADRB2 1451/4885SLC6A3 4750/4885
US-20230094341-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF HSD17B3, HSD17B11, HSD17B1 SLC6A4 2816/4885ADRB2 1854/4885SLC6A3 2221/4885
US-11236095-B2 Protein kinase B inhibitors PRKAR2B, PRKCB, AKT1 SLC6A4 4654/4885ADRB2 1451/4885SLC6A3 4750/4885
US-11760760-B2 Protein kinase B inhibitors PRKAR2B, PRKCB, AKT1 SLC6A4 4654/4885ADRB2 1451/4885SLC6A3 4750/4885
US-11957687-B2 Modulators of HSD17B13 and methods of use thereof HSD17B3, HSD17B11, HSD17B1 SLC6A4 2816/4885ADRB2 1854/4885SLC6A3 2221/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.