SCHEMBL3913657

SCHEMBL3913657

CN(CCCNC(=O)[C@H](CC1CCCCC1)NC(=O)O)C(=O)OC(C)(C)C

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.53
CTSK P43235 2/20 0.53
MMP2 P08253 9/20 0.43
MMP1 P03956 8/20 0.43
MMP3 P08254 8/20 0.43
CHRNB2 P17787 7/20 0.42
CHRNB4 P30926 7/20 0.42
CHRNA3 P32297 7/20 0.42
CHRNA4 P43681 7/20 0.42
GRIN1 Q05586 3/20 0.42
GRIN2A Q12879 3/20 0.42
GRM1 Q13255 3/20 0.42
CPB2 Q96IY4 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14360835 0.85 CTSS (0.55) CTSSCTSKMMP2MMP1MMP3
SCHEMBL14360791 0.84 METAP2 (0.43) CTSSCTSKMMP2MMP1MMP3
SCHEMBL14360790 0.79 TACR2 (0.49) CTSSCTSKCHRNB2CHRNB4CHRNA3
SCHEMBL3915529 0.77 BCHE (0.42) MMP2MMP1MMP3
SCHEMBL1864993 0.77 CHRNB2 (0.61) CTSSCTSKMMP1MMP3CHRNB2
SCHEMBL1861306 0.76 CTSK (0.69) CTSSCTSKCHRNB2CHRNB4CHRNA3
SCHEMBL1861303 0.76 CTSK (0.69) CTSSCTSKCHRNB2CHRNB4CHRNA3
SCHEMBL13739944 0.75 CHRNB2 (0.49) CTSSCTSKMMP2MMP1MMP3
SCHEMBL31040440 0.74 CA14 (0.50) CTSK
SCHEMBL4971388 0.71 CTSS (0.52) CTSSCTSKCHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797065-A4 ACYCLIC 1,3-DIAMINES AND USES THEREFOR SMITHKLINE BEECHAM CORP (US) 2009-03-04 EP disclosed
EP-1797065-A2 ACYCLIC 1,3-DIAMINES AND USES THEREFOR SMITHKLINE BEECHAM CORPORATION (US) 2007-06-20 EP disclosed
WO-2006029210-A2 ACYCLIC 1,3-DIAMINES AND USES THEREFOR SMITHKLINE BEECHAM CORPORATION (US) 2006-03-16 WO disclosed