SCHEMBL3922008

SCHEMBL3922008

CCOC(=O)C(F)Cc1ccc(O)cc1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.53
ESR2 Q92731 6/20 0.53
CA12 O43570 2/20 0.49
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA7 P43166 2/20 0.49
CA9 Q16790 2/20 0.49
CA14 Q9ULX7 2/20 0.49
PTGS2 P35354 3/20 0.46
MIF P14174 1/20 0.46
BACE1 P56817 1/20 0.43
SLC7A5 Q01650 1/20 0.43
TAAR1 Q96RJ0 3/20 0.43
SLC6A2 P23975 1/20 0.43
MMP8 P22894 1/20 0.42
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5305730 0.86 ESR1 (0.65) ESR1ESR2MIFSLC7A5TAAR1
SCHEMBL14541013 0.86 ESR1 (0.65) ESR1ESR2MIFSLC7A5TAAR1
SCHEMBL3629843 0.85 LMNA (0.50) MMP8KMT2A
SCHEMBL8870407 0.84 MMP8 (0.58) MMP8KMT2A
SCHEMBL5800254 0.82 MMP8 (0.55) ESR1ESR2CA12CA1CA2
SCHEMBL3694538 0.81 ESR1 (0.51) ESR1ESR2CA12CA1CA2
SCHEMBL5360147 0.81 ESR1 (0.51) ESR1ESR2CA12CA1CA2
SCHEMBL5385979 0.81 ESR1 (0.50) ESR1ESR2CA12CA1CA2
SCHEMBL13715359 0.81 ESR1 (0.50) ESR1ESR2CA12CA1CA2
SCHEMBL13715362 0.81 ESR1 (0.50) ESR1ESR2CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1698624-B1 PHENYLPROPANOIC ACID DERIVATIVES TAKEDA PHARMACEUTICAL (JP) 2012-06-27 EP disclosed
US-7585880-B2 Phenylpropanoic acid derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-09-08 US disclosed
US-7585880-B2 Phenylpropanoic acid derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-09-08 US disclosed
US-7585880-B2 Phenylpropanoic acid derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-09-08 US disclosed
US-20070155808-A1 Phenylpropanoic acid derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-07-05 US disclosed
US-20070155808-A1 Phenylpropanoic acid derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-07-05 US disclosed
US-20070155808-A1 Phenylpropanoic acid derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-07-05 US disclosed
EP-1698624-A1 PHENYLPROPANOIC ACID DERIVATIVES Takeda Pharmaceutical Company Limited (JP) 2006-09-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070155808-A1 Phenylpropanoic acid derivatives GPR119, GPR55, FFAR1 ESR1 317/4885ESR2 1025/4885CA12 4405/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.