SCHEMBL3926249

SCHEMBL3926249

CC(=O)Nc1ccc(S(=O)(=O)Nc2cccc(C)n2)cc1

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.66
ALDH1A1 P00352 3/20 0.65
HPGD P15428 2/20 0.65
HSD17B10 Q99714 2/20 0.65
L3MBTL1 Q9Y468 2/20 0.64
HSD11B1 P28845 6/20 0.63
ATIC P31939 1/20 0.60
LMNA P02545 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10031589 0.87 KDM4E (0.59) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL10031565 0.85 KDM4E (0.59) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL10031601 0.82 KDM4E (0.55) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL3486583 0.81 HSD11B1 (0.91) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL29506329 0.81 HSD11B1 (0.91) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL547543 0.80 KDM4E (1.00) KDM4EALDH1A1L3MBTL1ATIC
SCHEMBL29967633 0.79 KDM4E (1.00) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL6026817 0.79 KDM4E (1.00) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL29776905 0.79 TSHR (0.73) ALDH1A1L3MBTL1LMNA
SCHEMBL6027289 0.79 ALDH1A1 (0.74) KDM4EALDH1A1HPGDHSD17B10L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8110338-B2 Heat-sensitive positive-working lithographic printing plate precursor AGFA GRAPHICS NV (BE) 2012-02-07 US disclosed
US-8110338-B2 Heat-sensitive positive-working lithographic printing plate precursor AGFA GRAPHICS NV (BE) 2012-02-07 US disclosed
US-20090170028-A1 HEAT-SENSITIVE POSITIVE-WORKING LITHOGRAPHIC PRINTING PLATE PRECURSOR AGFA GRAPHICS NV (BE) 2009-07-02 US disclosed
US-20090170028-A1 HEAT-SENSITIVE POSITIVE-WORKING LITHOGRAPHIC PRINTING PLATE PRECURSOR AGFA GRAPHICS NV (BE) 2009-07-02 US disclosed
US-7482341-B2 N-(pyridin-2-yl)-benzenesulfonamides; antidiabetic agents for Type II Diabetes; obesity; 11beta-hydroxysteroid dehydrogenase inhibitors HOFFMANN-LA ROCHE INC. (US) 2009-01-27 US disclosed
WO-2007099047-A1 A HEAT-SENSITIVE POSITIVE-WORKING LITHOGRAPHIC PRINTING PLATE PRECURSOR AGFA GRAPHICS NV (BE) 2007-09-07 WO disclosed
EP-1826001-A1 A heat-sensitive positive-working lithographic printing plate precursor Agfa Graphics N.V. (BE) 2007-08-29 EP disclosed
WO-2006037501-A9 ALKIL-PYRIDINES AS 11-BETA INHIBITORS FOR DIABETES HOFFMANN LA ROCHE (CH) 2007-08-02 WO disclosed
EP-1799647-A1 ALKIL-PYRIDINES AS 11-BETA INHIBITORS FOR DIABETES F.HOFFMANN-LA ROCHE AG (CH) 2007-06-27 EP disclosed
WO-2006037501-A1 ALKIL-PYRIDINES AS 11-BETA INHIBITORS FOR DIABETES F. HOFFMANN-LA ROCHE AG (CH) 2006-04-13 WO disclosed
US-20060074237-A1 N-(pyridin-2-yl)-benzenesulfonamides; hypotensive agents; antidiabetic agents for Type II Diabetes; obesity, eating disorders, dyslipidemia; 11beta-hydroxysteroid dehydrogenase inhibitors HOFFMANN-LA ROCHE INC. 2006-04-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060074237-A1 N-(pyridin-2-yl)-benzenesulfonamides; hypotensive agents; antidiabetic agents for Type II Diabetes; obesity, eating disorders, dyslipidemia; 11beta-hydroxysteroid dehydrogenase inhibitors HSD3B1, HSD3B2, HSD11B2 KDM4E 1422/4885ALDH1A1 210/4885HPGD 147/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.