SCHEMBL3926529

SCHEMBL3926529

C[Si](C)(C)CCOCn1cc2cc(C(F)(F)F)cc(CCO)c2n1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
DGAT1 O75907 4/20 0.35
ALOX5AP P20292 1/20 0.31
FEN1 P39748 1/20 0.31
GPR52 Q9Y2T5 1/20 0.30
S1PR1 P21453 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3928026 0.89 DGAT1 (0.36) DGAT1ALOX5APFEN1
SCHEMBL3935157 0.86 DGAT1 (0.33) DGAT1
SCHEMBL3936612 0.83 DGAT1 (0.30) DGAT1
SCHEMBL3925961 0.82 MEN1 (0.30) DGAT1
SCHEMBL2428508 0.80 DGAT1 (0.34) DGAT1ALOX5APFEN1S1PR1
SCHEMBL2428806 0.79 DGAT1 (0.35) DGAT1ALOX5APFEN1S1PR1
SCHEMBL2430892 0.78 DGAT1 (0.36) DGAT1ALOX5APFEN1
SCHEMBL3923489 0.77 DGAT1 (0.38) IDO1TDO2DGAT1ALOX5APFEN1
SCHEMBL3936516 0.76 TACR1 (0.46)
SCHEMBL3926165 0.74 TACR1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009009411-A1 SUBSTITUTED HETEROCYCLIC ETHERS AND THEIR USE IN CNS DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-15 WO disclosed