SCHEMBL39270

SCHEMBL39270

C=CCNc1nc(-c2cc(Cl)ccc2Cl)cs1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.67
RAB9A P51151 6/20 0.67
MAPT P10636 6/20 0.67
SMN1; SMN2 Q16637 5/20 0.67
MEN1 O00255 4/20 0.67
KMT2A Q03164 4/20 0.67
NFKB1 P19838 2/20 0.67
NFKB2 Q00653 2/20 0.67
RELA Q04206 2/20 0.67
CYP1A2 P05177 1/20 0.67
CYP3A4 P08684 1/20 0.67
CYP2D6 P10635 1/20 0.67
CYP2C9 P11712 1/20 0.67
CYP2C19 P33261 1/20 0.67
PKM P14618 1/20 0.54
RORC P51449 9/20 0.54
ALDH1A1 P00352 3/20 0.53
HPGD P15428 2/20 0.53
KDM4E B2RXH2 2/20 0.51
TP53 P04637 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL37686 0.84 NPC1 (0.63) NPC1RAB9AMAPTSMN1; SMN2MEN1
SCHEMBL14814817 0.77 PKM (0.61) MAPTSMN1; SMN2MEN1KMT2ACYP1A2
SCHEMBL1916174 0.77 PKM (0.65) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL37919 0.73 MAPT (0.56) NPC1RAB9AMAPTSMN1; SMN2MEN1
SCHEMBL1915688 0.73 PKM (0.56) NPC1RAB9APKMRORCHPGD
SCHEMBL3598222 0.72 PKM (0.65) MAPTCYP1A2PKMRORCHPGD
SCHEMBL1916623 0.72 RORC (0.58) NPC1RAB9AMAPTSMN1; SMN2MEN1
SCHEMBL38629 0.72 MAPT (0.74) NPC1RAB9AMAPTSMN1; SMN2MEN1
SCHEMBL38117 0.71 GSTO1 (0.58) NPC1RAB9AMAPTSMN1; SMN2MEN1
SCHEMBL1800878 0.70 ALDH1A1 (0.65) PKMRORCALDH1A1KDM4EAMY1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011151436-A2 NOVEL COMPOUNDS, METHOD FOR USE THEM AND PHARMACEUTICAL COMPOSITION CONTAINING THEM EUROSCREEN S.A. (BE) 2011-12-08 WO disclosed