SCHEMBL3930680

SCHEMBL3930680

CCC1=N[C@@H](C(=O)O)CS1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 8/20 0.38
GABRB2 P47870 8/20 0.38
GABRA1 P14867 6/20 0.38
GABRR1 P24046 6/20 0.38
GABRA4 P48169 4/20 0.38
SLC6A12 P48065 1/20 0.38
SLC6A13 Q9NSD5 1/20 0.38
GPR35 Q9HC97 1/20 0.35
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9885411 1.00 GABRA5 (0.38) GABRA5GABRB2GABRA1GABRR1GABRA4
SCHEMBL13547558 0.86 GABRA1 (0.33) GABRA5GABRB2GABRA1GABRR1GABRA4
SCHEMBL7033502 0.82 GABRA1 (0.33) GABRA5GABRB2GABRA1GABRR1GABRA4
SCHEMBL19627500 0.82 KMT2A (0.34) GABRA5GABRB2GABRA1GABRR1GABRA4
SCHEMBL10716460 0.81 GPR35 (0.34) GABRA5GABRB2GABRA1GABRR1GABRA4
SCHEMBL7012526 0.76 GPR35 (0.33) GABRA5GABRB2GABRA1GABRR1GABRA4
SCHEMBL12835928 0.75
SCHEMBL22493427 0.75
SCHEMBL19884781 0.75
SCHEMBL14660290 0.74 MAPT (0.36) GABRA5GABRB2GABRA1GABRR1GABRA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346026-B1 MICROORGANISM PRODUCING 5'-INOSINIC ACID AND PROCESS FOR PRODUCING 5'-INOSINIC ACID USING THE SAME CJ CHEILJEDANG CORP (KR) 2009-04-01 EP claimed
US-7244608-B2 Microorganism producing 5′-inosinic acid and process for producing 5′-inosinic acid using the same CHEIL JEDANG CORPORATION (KR) 2007-07-17 US claimed
EP-1346026-A4 MICROORGANISM PRODUCING 5'-INOSINIC ACID AND PROCESS FOR PRODUCING 5'-INOSINIC ACID USING THE SAME CHEIL JEDANG CORP (KR) 2004-06-23 EP claimed
EP-1346026-A1 MICROORGANISM PRODUCING 5'-INOSINIC ACID AND PROCESS FOR PRODUCING 5'-INOSINIC ACID USING THE SAME Cheil Jedang Corporation (KR) 2003-09-24 EP claimed
US-20030054504-A1 Microorganism producing 5'-inosinic acid and process for producing 5'-inosinic acid using the same CJ CHEILJEDANG CORPORATION (KP) 2003-03-20 US claimed
WO-2002051984-A1 MICROORGANISM PRODUCING 5'-INOSINIC ACID AND PROCESS FOR PRODUCING 5'-INOSINIC ACID USING THE SAME CHEIL JEDANG CORPORATION (KR) 2002-07-04 WO claimed
EP-3290413-B9 PYRIDINONE AND PYRIMIDINONE DERIVATIVES AS FACTOR XIA INHIBITORS ONO PHARMACEUTICAL CO (JP) 2020-04-29 EP disclosed
EP-3290413-B1 PYRIDINONE AND PYRIMIDINONE DERIVATIVES AS FACTOR XIA INHIBITORS ONO PHARMACEUTICAL CO (JP) 2019-11-13 EP disclosed
EP-1346026-B1 MICROORGANISM PRODUCING 5'-INOSINIC ACID AND PROCESS FOR PRODUCING 5'-INOSINIC ACID USING THE SAME CJ CHEILJEDANG CORP (KR) 2009-04-01 EP disclosed
US-7244608-B2 Microorganism producing 5′-inosinic acid and process for producing 5′-inosinic acid using the same CHEIL JEDANG CORPORATION (KR) 2007-07-17 US disclosed
EP-1346026-A4 MICROORGANISM PRODUCING 5'-INOSINIC ACID AND PROCESS FOR PRODUCING 5'-INOSINIC ACID USING THE SAME CHEIL JEDANG CORP (KR) 2004-06-23 EP disclosed
EP-1346026-A1 MICROORGANISM PRODUCING 5'-INOSINIC ACID AND PROCESS FOR PRODUCING 5'-INOSINIC ACID USING THE SAME Cheil Jedang Corporation (KR) 2003-09-24 EP disclosed
US-20030054504-A1 Microorganism producing 5'-inosinic acid and process for producing 5'-inosinic acid using the same CJ CHEILJEDANG CORPORATION (KP) 2003-03-20 US disclosed
WO-2002051984-A1 MICROORGANISM PRODUCING 5'-INOSINIC ACID AND PROCESS FOR PRODUCING 5'-INOSINIC ACID USING THE SAME CHEIL JEDANG CORPORATION (KR) 2002-07-04 WO disclosed