SCHEMBL3931209

SCHEMBL3931209

CS(=O)(=O)c1ccc(N(CCN2CCC(C(=O)O)CC2)c2cccc(F)c2)cc1.N#Cc1ccc(CN)cc1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 11/20 0.42
KCNH2 Q12809 8/20 0.39
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
DRD2 P14416 1/20 0.38
HRH1 P35367 1/20 0.38
TAS2R14 Q9NYV8 1/20 0.37
CCR2 P41597 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3931201 0.87 CCR5 (0.52) CCR5KCNH2
SCHEMBL3928869 0.79 CCR5 (0.48) CCR5
SCHEMBL13929221 0.77 SIGMAR1 (0.48) CCR5KCNH2
SCHEMBL13929220 0.76 SIGMAR1 (0.56) CCR5
SCHEMBL3931205 0.74 OPRM1 (0.40) CCR5KCNH2CCR2
SCHEMBL4260236 0.73 MAPT (0.49) CCR5DRD2
SCHEMBL13930630 0.73 MAPT (0.49) CCR5KCNH2CCR2
SCHEMBL3931152 0.69 LTA4H (0.50) HTR2A
SCHEMBL4217001 0.66 SIGMAR1 (0.57) CCR5
SCHEMBL4771551 0.66 CCR5 (0.77) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009010480-A1 1-{2-[(DIPHENYL)AMINO]-ETHYL}-PIPERIDINE-4-CARBOXYLIC ACID BENZYLAMIDE DERIVATIVES AND RELATED COMPOUNDS AS CCR5 AGONISTS FOR THE TREATMENT OF IMMUNE AND INFLAMMATORY DISEASES EUROSCREEN S.A. (BE) 2009-01-22 WO disclosed